IP Library Granted Patent US 9,505,842
Granted Patent B2
US 9,505,842 · App. 14/509,353 · Granted Nov 29, 2016

Methods for inhibiting the binding of endosialin to ligands

Inventors: Yuhong Zhou (Phoenixville, PA); Brian Tomkowicz (East Norriton, PA); Luigi Grasso (Bryn Mawr, PA); Nicholas C. Nicolaides (Glen Mills, PA); Philip M. Sass (Audubon, PA)
Assignee: Morphotek, Inc.
C07K16/2851A61K2039/505C07K2316/96C07K2317/14C07K2317/24C07K2317/56C07K2317/76C07K2319/30
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Quick Facts
Patent No.
US 9,505,842
App. No.
14/509,353
Granted
Nov 29, 2016
Kind
B2
Abstract

The invention provides methods for inhibiting the interaction of endosialin with endosialin ligands. The inhibition is effectuated on the genetic level, by inhibiting endosialin gene expression, and on the protein level, by blocking the interaction of cell-surface expressed endosialin with ligands such as fibronectin and collagen. The invention provides methods for identifying inhibitors of the interaction of endosialin with endosialin ligands. Also provided are methods for inhibiting angiogenesis and neovascularization in vivo and in vitro.

Claims (5)

1. A monoclonal antibody or antigen-binding fragment thereof that specifically binds endosialin, said antibody or antigen-binding fragment produced by cells having ATCC Access. No. PTA-9017.

2. The antibody or antigen-binding fragment of claim 1 comprising a detectable label.

3. The antibody or antigen-binding fragment of claim 2 wherein said detectable label comprises a fluorescent label, a radiolabel, or biotin.

4. The antibody or antigen-binding fragment of claim 1 conjugated to a cytotoxin.

5. The antibody or antigen-binding fragment of claim 4 , wherein said cytotoxin comprises a bacterial toxin, a viral toxin, or a radioisotope.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 5, 2018
From: MORPHOTEK, INC.
To: EISAI, INC.
Reel/Frame 046498/0446 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 21, 2018
From: ZHOU, YUHONG; TOMKOWICZ, BRIAN; GRASSO, LUIGI; NICOLAIDES, NICHOLAS C.; SASS, PHILIP M.
To: MORPHOTEK, INC.
Reel/Frame 046166/0909 →
Continuity (5)
Continuation 12873667 · Sep 1, 2010
Continuation 12062630 · Apr 4, 2008
Provisional Application 60910362 · Apr 5, 2007
Provisional Application 60980026 · Oct 15, 2007
Related Publication 20150079104A1 · Mar 19, 2015