IP Library Granted Patent US 10,155,813
Granted Patent B2
US 10,155,813 · App. 15/098,627 · Granted Dec 18, 2018

Fully human antibodies to BTLA

Inventors: Jennifer Marie Mataraza (Cambridge, MA); Andrea Van Elsas (Oss, NL); Alan J. Korman (Piedmont, CA); Edward L. Halk (Sunnyvale, CA); Kent B. Thudium (Oakland, CA); Mark J. Selby (San Francisco, CA); Timothy W. Sproul (Livermore, CA); Heidi N. Leblanc (Mountain View, CA)
Assignee: E. R. Squibb & Sons, L.L.C.
C07K16/2803C07K16/2818A61K2039/505C07K2317/21C07K2317/24C07K2317/56C07K2317/565C07K2317/73C07K2317/77C07K2317/92
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Quick Facts
Patent No.
US 10,155,813
App. No.
15/098,627
Granted
Dec 18, 2018
Kind
B2
Abstract

The present invention relates to binding compounds specific for BTLA and uses thereof. More specifically, the invention relates to fully human antibodies that recognize human BTLA and modulate its activity in cancer, inflammatory, and autoimmune disorders.

Claims (4)

1. A method of treating cancer in a subject comprising administering an effective amount of an antibody, or antigen binding fragment, comprising a heavy chain variable region CDR1 comprising the amino acid sequence of SEQ ID NO:19, a heavy chain variable region CDR2 comprising the amino acid sequence of SEQ ID NO:20, a heavy chain variable region CDR3 comprising the amino acid sequence of SEQ ID NO:21, a light chain variable region CDR1 comprising the amino acid sequence of SEQ ID NO:26, a light chain variable region CDR2 comprising the amino acid sequence of SEQ ID NO:27; and a light chain variable region CDR3 comprising the amino acid sequence of SEQ ID NO:28, wherein the antibody, or antigen binding fragment, specifically binds human BTLA.

2. The method of claim 1 , wherein the cancer is selected from the group consisting of melanoma, renal cancer, prostate cancer, pancreatic adenocarcinoma, breast cancer, colon cancer, lung cancer, esophageal cancer, squamous cell carcinoma of the head and neck, liver cancer, ovarian cancer, cervical cancer, thyroid cancer, glioblastoma, glioma, leukemia, lymphoma, and neoplastic malignancies.

3. A method of treating cancer in a subject comprising administering an effective amount of an antibody, or antigen binding fragment, comprising heavy and light chain variable regions as set forth in SEQ ID NOs:25 and 32, respectively, wherein the antibody, or antigen binding fragment, specifically binds human BTLA.

4. The method of claim 3 , wherein the cancer is selected from the group consisting of melanoma, renal cancer, prostate cancer, pancreatic adenocarcinoma, breast cancer, colon cancer, lung cancer, esophageal cancer, squamous cell carcinoma of the head and neck, liver cancer, ovarian cancer, cervical cancer, thyroid cancer, glioblastoma, glioma, leukemia, lymphoma, and neoplastic malignancies.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 28, 2016
From: KORMAN, ALAN J.; HALK, EDWARD L.; THUDIUM, KENT B.; SELBY, MARK; SPROUL, TIMOTHY W.; LEBLANC, HEIDI N.
To: MEDAREX, INC.
Reel/Frame 038412/0726 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 28, 2016
From: MATARAZA, JENNIFER MARIE; ELSAS, ANDREA VAN
To: N.V. ORGANON
Reel/Frame 038412/0770 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 28, 2016
From: N.V. ORGANON
To: MEDAREX, INC.
Reel/Frame 038412/0809 →
MERGER Recorded Apr 28, 2016
From: MEDAREX, L.L.C.
To: E.R. SQUIBB & SONS, L.L.C.
Reel/Frame 038412/0871 →
MERGER Recorded Apr 28, 2016
From: MEDAREX, INC.
To: MEDAREX, L.L.C.
Reel/Frame 038556/0590 →
Continuity (5)
Division 14031319 · Sep 19, 2013
Division 13388028
Provisional Application 61257612 · Nov 3, 2009
Provisional Application 61230332 · Jul 31, 2009
Related Publication 20160222114A1 · Aug 4, 2016