IP Library › Granted Patent US 10,245,267
Granted Patent B2
US 10,245,267 · App. 15/601,423 · Granted Apr 2, 2019

Biaryl amide compounds as kinase inhibitors

Inventors: Robert John Aversa (Cambridge, MA); Paul Andrew Barsanti (Pleasant Hill, CA); Matthew T. Burger (Cambridge, MA); Michael Patrick Dillon (Cambridge, MA); Alan Dipesa (Bronx, NY); Cheng Hu (San Mateo, CA); Yan Lou (Pleasanton, CA); Gisele A. Nishiguchi (Cambridge, MA); Yue Pan (Cambridge, MA); Valery Rostislavovich Polyakov (Emeryville, CA); Savithri Ramurthy (Cambridge, MA); Alice C. Rico (Emeryville, CA); Lina Quattrocchio Setti (Fremont, CA); Aaron Smith (Emeryville, CA); Sharadha Subramanian (Emeryville, CA); Benjamin R. Taft (Emeryville, CA); Huw Roland Tanner (San Francisco, CA); Lifeng Wan (Emeryville, CA); Naeem Yusuff (Cambridge, MA)
Assignee: Novartis AG
A61K31/5377A61K31/444A61K31/501A61K31/5375A61K31/541A61K45/06C07B59/002C07D213/74C07D213/75C07D213/81C07D213/82C07D213/84C07D233/88C07D237/20C07D237/22C07D237/24C07D239/42C07D239/47C07D239/48C07D241/20C07D263/58C07D277/42C07D401/04C07D401/12C07D401/14C07D403/04C07D403/12C07D405/04C07D405/12C07D405/14C07D409/14C07D413/04C07D413/12C07D413/14C07D417/12C07D471/04C07D487/04C07D491/04C07D491/048C07D491/08C07D491/107C07D493/04C07D493/10C07D495/04C07D498/08C07D513/04C07B2200/05
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Quick Facts
Patent No.
US 10,245,267
App. No.
15/601,423
Granted
Apr 2, 2019
Kind
B2
Abstract

The present invention provides compounds of Formula (I) as described herein, and salts thereof, and therapeutic uses of these compounds for treatment of disorders associated with Raf kinase activity. The invention further provides pharmaceutical compositions comprising these compounds, and compositions comprising these compounds and a therapeutic co-agent.

Claims (4)

1. A compound, or a pharmaceutically acceptable salt thereof, selected from:

2. A pharmaceutical composition comprising a compound of claim 1 or a pharmaceutically acceptable salt thereof and one or more pharmaceutically acceptable carriers.

3. A combination comprising a therapeutically effective amount of a compound according to claim 1 or a pharmaceutically acceptable salt thereof and one or more therapeutically active co-agents.

4. A method of treating a proliferative disorder selected from non-small cell lung cancer and ovarian cancer, comprising administering to a subject having said disorder a therapeutically effective amount of a compound of claim 1 or a pharmaceutically acceptable salt thereof.

Assignments (6)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 14, 2017
From: YUSUFF, NAEEM
To: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC.
Reel/Frame 043585/0589 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 14, 2017
From: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC.
To: NOVARTIS AG
Reel/Frame 043585/0739 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 14, 2017
From: DIPESA, ALAN
To: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC.
Reel/Frame 043585/0791 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 14, 2017
From: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC.
To: NOVARTIS AG
Reel/Frame 043585/0828 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 14, 2017
From: NOVARTIS VACCINES AND DIAGNOSTICS, INC.
To: NOVARTIS AG
Reel/Frame 043586/0353 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 14, 2017
From: ROBERT AVERSA; BARSANTI, PAUL A.; BURGER, MATTHEW; DILLON, MICHAEL PATRICK; HU, CHENG; LOU, YAN; NISHIGUCHI, GISELE; PAN, YUE; POLYAKOV, VALERY; RAMURTHY, SAVITHRI; RICO, ALICE; SETTI, LINA; SMITH, AARON; SUBRAMANIAN, SHARADHA; TAFT, BENJAMIN; TANNER, HUW; WAN, LIFENG
To: NOVARTIS VACCINES AND DIAGNOSTICS, INC.
Reel/Frame 043859/0857 →
Continuity (3)
Division 14774431
Provisional Application 61783558 · Mar 14, 2013
Related Publication 20170260207A1 · Sep 14, 2017
Cited By (1)
US 12,187,703