IP Library › Granted Patent US 10,342,763
Granted Patent B2
US 10,342,763 · App. 15/831,866 · Granted Jul 9, 2019

Chewable soft capsules

Inventors: EmadEldin M. Hassan (Parkton, MD); Warren Walter Kindt (Ossineke, MI); Roger E. Gordon (Stokesdale, NC)
Assignee: Patheon Softgels, Inc.
A61K9/4816A61K9/0056A61K9/4825A61K9/4858A61K9/4866A61K31/135A61K31/137A61K31/167A61K31/19A61K31/192
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Quick Facts
Patent No.
US 10,342,763
App. No.
15/831,866
Granted
Jul 9, 2019
Kind
B2
Abstract

A matrix formulation for a soft chewable capsule is provided which includes a gel-forming composition, a plasticizer, a polymer modifier, and water. The polymer modifier may be a carboxylic acid or other organic compound that alters the physical and/or chemical properties of the capsule formulation. A chewable soft capsule is also provided, having enhanced organoleptic and processing properties. An active material may be delivered to a user using this dosage form. A method of forming the chewable soft capsule is also provided.

Claims (53)

1. A soft capsule suitable for chewing or buccal dissolution comprising

a sheath encapsulating a matrix,

the sheath comprising:

one or more gel-forming polymers;

one or more plasticizers;

one or more polymer modifiers comprising a carboxylic acid; and

water; and

the matrix comprising:

one or more second gel-forming polymers;

one or more non-steroidal anti-inflammatory drugs (NSAIDs); and

water.

2. The soft capsule of claim 1 , wherein the gel-forming polymer comprises gelatin, partially hydrolyzed gelatin, hydrolyzed gelatin, or a combination thereof.

3. The soft capsule of claim 1 , wherein the plasticizer comprises maltitol, glycerin, xylitol, or a combination thereof.

4. The soft capsule of claim 1 , wherein the polymer modifier comprises citric acid, lactic acid, tartaric acid, fumaric acid, glycolic acid, or a combination thereof.

5. The soft capsule of claim 1 , wherein the polymer modifier comprises citric acid.

6. The soft capsule of claim 1 , wherein the second gel-forming polymer comprises gelatin, partially hydrolyzed gelatin, hydrolyzed gelatin, or a combination thereof.

7. The soft capsule of claim 1 , wherein non-steroidal anti-inflammatory drug comprises ibuprofen, naproxen, celecoxib, or aspirin.

8. The soft capsule of claim 1 , wherein the shell further comprises one or more of sweeteners, flavors, or colors.

9. The soft capsule of claim 1 , wherein the matrix further comprises one or more of sweeteners or flavors.

10. A soft capsule suitable for chewing or buccal dissolution comprising

a sheath encapsulating a matrix,

the sheath comprising:

one or more gel-forming polymers;

one or more plasticizers;

one or more polymer modifiers comprising a carboxylic acid; and

water; and

the matrix comprising:

one or more second gel-forming polymers;

ibuprofen; and

water.

11. The soft capsule of claim 10 , wherein the gel-forming polymer comprises gelatin, partially hydrolyzed gelatin, hydrolyzed gelatin, or a combination thereof.

12. The soft capsule of claim 10 , wherein the plasticizer comprises maltitol, glycerin, xylitol, or a combination thereof.

13. The soft capsule of claim 10 , wherein the polymer modifier comprises citric acid, lactic acid, tartaric acid, fumaric acid, glycolic acid, or a combination thereof.

14. The soft capsule of claim 10 , wherein the polymer modifier comprises citric acid.

15. The soft capsule of claim 10 , wherein the second gel-forming polymer comprises gelatin, partially hydrolyzed gelatin, hydrolyzed gelatin, or a combination thereof.

16. The soft capsule of claim 10 , wherein the shell further comprises one or more of sweeteners, flavors, or colors.

17. The soft capsule of claim 10 , wherein the matrix further comprises one or more of sweeteners or flavors.

18. A soft capsule suitable for chewing or buccal dissolution comprising

a sheath encapsulating a matrix,

the sheath comprising:

one or more gel-forming polymers;

one or more plasticizer;

one or more polymer modifiers comprising a carboxylic acid;

one or more sweeteners;

one or more flavors;

one or more colors; and

water; and

the matrix comprising:

one or more second gel-forming polymers;

one or more sweeteners;

one or more flavors;

ibuprofen; and

water.

Continuity (7)
Continuation 15590369 · May 9, 2017
Continuation 14790624 · Jul 2, 2015
Continuation 14316831 · Jun 27, 2014
Continuation 13327293 · Dec 15, 2011
Division 10512318
Provisional Application 60375479 · Apr 25, 2002
Related Publication 20180092853A1 · Apr 5, 2018