IP Library › Granted Patent US 10,799,487
Granted Patent B2
US 10,799,487 · App. 16/393,774 · Granted Oct 13, 2020

Compositions for the treatment of hypertension

Inventors: Anthony Rodgers (Newtown, AU); Stephen MacMahon (Newtown, AU)
Assignee: THE GEORGE INSTITUTE FOR GLOBAL HEALTH
A61K31/4422A61K31/277A61K31/382A61K31/40A61K31/404A61K31/4035A61K31/41A61K31/4178A61K31/4184A61K31/4418A61K31/495A61K31/517A61K31/549A61K31/554A61P9/12
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Quick Facts
Patent No.
US 10,799,487
App. No.
16/393,774
Filed
Apr 24, 2019
Granted
Oct 13, 2020
Kind
B2
Art Unit
1627
USPC
514/356
Abstract

Provided herein are pharmaceutical compositions that are useful for the treatment of hypertension comprising an angiotensin II receptor blocker, a diuretic, and a calcium channel blocker.

Claims (24)

1. A pharmaceutical composition comprising:

(a) telmisartan;

(b) indapamide; and

(c) amlodipine besylate;

wherein a dose of telmisartan is from about 16 mg to about 24 mg, a dose of indapamide is from about 1 mg to about 1.5 mg, and a dose of amlodipine besylate is from about 2 mg to about 3 mg; and wherein the pharmaceutical composition is free of a beta-blocker.

2. The pharmaceutical composition of claim 1 , wherein the dose of indapamide is about 1.25 mg.

3. The pharmaceutical composition of claim 1 , wherein the dose of amlodipine besylate is about 2.5 mg.

4. The pharmaceutical composition of claim 1 , wherein the dose of telmisartan is about 20 mg.

5. The pharmaceutical composition of claim 1 , wherein the dose of indapamide is about 1.25 mg and the dose of amlodipine besylate is about 2.5 mg.

6. The pharmaceutical composition of claim 1 , wherein the dose of indapamide is about 1.25 mg and the dose of telmisartan is about 20 mg.

7. The pharmaceutical composition of claim 1 , wherein the dose of amlodipine besylate is about 2.5 mg and the dose of telmisartan is about 20 mg.

8. The pharmaceutical composition of claim 1 , wherein the dose of indapamide is about 1.25 mg, the dose of amlodipine besylate is about 2.5 mg, and the dose of telmisartan is about 20 mg.

9. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is suitable for oral administration.

10. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is in the form of pill, tablet, or capsule.

11. A method of treating hypertension in a subject in need thereof comprising administering to the subject the pharmaceutical composition of claim 1 .

12. The method of claim 11 , wherein the treatment results in a systolic blood pressure (SBP) of less than about 140 mmHg.

13. The method of claim 11 , wherein the treatment results in a reduction of systolic blood pressure (SBP) of about 10 mmHg or greater.

14. The method of claim 11 , wherein the treatment results in a diastolic blood pressure (DBP) of less than about 90 mmHg.

15. The method of claim 11 , wherein the treatment results in a reduction of diastolic blood pressure (DBP) of about 5 mmHg or greater.

16. The method of claim 11 , wherein treatment results in a reduction in systolic blood pressure (SBP) that is greater than the reduction obtained with the full lowest hypertension therapeutic dose of any one of the (a), (b), and (c) in the pharmaceutical composition.

17. The method of any one of claim 11 , wherein treatment results in a reduction in diastolic blood pressure (DBP) that is greater than the reduction obtained with the full lowest hypertension therapeutic dose of any one of (a), (b), and (c) in the pharmaceutical composition.

18. The method of claim 11 , wherein the treatment results in greater long term tolerability and reduced risk of side effects when compared to treatment with the full lowest hypertension therapeutic dose of any one of (a), (b), and (c) in the pharmaceutical composition.

19. The method of claim 11 , wherein the treatment is the initial or first-line treatment of hypertension.

20. The method of claim 11 , wherein the subject has not received any previous hypertension therapy prior to treatment.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 24, 2019
From: RODGERS, ANTHONY; MACMAHON, STEPHEN
To: THE GEORGE INSTITUTE FOR GLOBAL HEALTH
Reel/Frame 048987/0145 →
Continuity (4)
Continuation 15919923 · Mar 13, 2018
Continuation PCTIB2018000083 · Jan 23, 2018
Provisional Application 62450324 · Jan 25, 2017
Related Publication 20190343818A1 · Nov 14, 2019
Cited By (5)
US 12,285,415 US 12,465,599 US 12,521,380 US 12,661,345 US 12,673,047