IP Library Granted Patent US 10,894,041
Granted Patent B2
US 10,894,041 · App. 16/275,669 · Granted Jan 19, 2021

Medical treatments based on anamorelin

Inventors: William Mann (Hoboken, NJ); John Friend (Colts Neck, NJ); William Polvino (Tinton Falls, NJ); Suzan Allen (Georgetown, TX); Ming Lu (Plainsboro, NJ); Elizabeth Duus (Cape Coral, FL); Ruben Giorgino (Allschwil, CH); Enrico Baroni (Cernobbio, IT)
Assignee: Helsinn Healthcare SA
A61K31/454A61K31/00
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Quick Facts
Patent No.
US 10,894,041
App. No.
16/275,669
Granted
Jan 19, 2021
Kind
B2
Abstract

Methods of treating cancer related conditions using anamorelin are described.

Claims (27)

1. A method of treating weight loss associated with cancer in a patient in need thereof comprising administering to said patient a therapeutically effective amount of anamorelin or a pharmaceutically acceptable salt thereof, wherein:

a) said patient has a body mass index of <20 kg/m 2 ; and

b) said patient has involuntary weight loss of >2% during the previous 6 months; and

said method increases the body weight of said patient.

2. The method of claim 1 , wherein said patient has an ECOG score of 0, 1, or 2.

3. The method of claim 1 , further for treating low quality of life as measured by FAACT in the anorexia/cachexia domain in said patient, wherein said patient has low quality of life as measured by FAACT in the anorexia/cachexia domain and said method improves said low quality of life.

4. The method of claim 1 , further for treating low quality of life as measured by FAACT in the anorexia/cachexia domain and low physical and functional well-being as measured by FAACT in the anorexia/cachexia domain in said patient, wherein:

a) said patient has low quality of life as measured by FAACT in the anorexia/cachexia domain; and

b) said patient has low physical and functional well-being as measured by FAACT in the anorexia/cachexia domain; and

said method improves said low quality of life and said low physical and functional well-being.

5. The method of claim 1 , wherein said patient has stage III unresectable or stage IV NSCLC.

6. The method of claim 1 , wherein said therapeutically effective amount comprises 100 mg of anamorelin or a pharmaceutically acceptable salt thereof once daily.

7. The method of claim 1 , wherein said therapeutically effective amount comprises 100 mg of anamorelin HCl based on the weight of the salt administered once daily.

8. The method of claim 4 , wherein said therapeutically effective amount comprises 100 mg of anamorelin or a pharmaceutically acceptable salt thereof once daily.

9. A method of treating weight loss associated with cancer, and anorexia symptoms as measured by FAACT in the anorexia/cachexia domain, in a patient in need thereof comprising administering to said patient a therapeutically effective amount of anamorelin or a pharmaceutically acceptable salt thereof, wherein:

a) said patient has a body mass index of <20 kg/m 2 ;

b) said patient has involuntary weight loss of >2% during the previous 6 months;

c) said method increases the body weight of said patient; and

d) said method improves said anorexia symptoms.

10. The method of claim 9 , wherein said patient has an ECOG score of 0, 1, or 2.

11. The method of claim 9 , further wherein said patient has low quality of life as measured by FAACT in the anorexia/cachexia domain and said method improves said quality of life.

12. The method of claim 9 , wherein said patient has stage III unresectable or stage IV NSCLC.

13. The method of claim 9 , wherein said therapeutically effective amount comprises 100 mg of anamorelin or a pharmaceutically acceptable salt thereof once daily.

14. The method of claim 9 , wherein said therapeutically effective amount comprises 100 mg of anamorelin HCl based on the weight of the salt administered once daily.

15. The method of claim 9 , wherein said patient has low physical and functional well-being as measured by FAACT in the anorexia/cachexia domain and said method improves said physical and functional well-being.

16. The method of claim 9 , wherein said improvement in anorexia symptoms is measured by a subset of FAACT in the anorexia/cachexia domain.

17. The method of claim 9 , wherein said improvement in anorexia symptoms is measured by the entire FAACT in the anorexia/cachexia domain.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 30, 2024
From: MANN, WILLIAM; FRIEND, JOHN; LU, MING; DUUS, ELIZABETH; POLVINO, WILLIAM; ALLEN, SUZAN; GIORGINO, RUBEN; BARONI, ENRICO
To: HELSINN HEALTHCARE SA
Reel/Frame 067575/0435 →
RELEASE OF SECURITY INTEREST Recorded Sep 20, 2023
From: HAMILTON SA LLC
To: HELSINN HEALTHCARE SA; HELSINN THERAPEUTICS (U.S.), INC.; HELSINN BIREX PHARMACEUTICALS LIMITED
Reel/Frame 064961/0567 →
SECURITY INTEREST Recorded Dec 30, 2022
From: HELSINN HEALTHCARE SA; HELSINN THERAPEUTICS (U.S.), INC.; HELSINN BIREX PHARMACEUTICALS LIMITED
To: HAMILTON SA LLC
Reel/Frame 062254/0888 →
Continuity (4)
Continuation 15590025 · May 9, 2017
Continuation 14839038 · Aug 28, 2015
Provisional Application 62045976 · Sep 4, 2014
Related Publication 20190175574A1 · Jun 13, 2019