IP Library Granted Patent US 11,660,309
Granted Patent B2
US 11,660,309 · App. 17/182,098 · Granted May 30, 2023

Prevention and treatment of inflammatory conditions

Inventor: Vipin Kumar Chaturvedi (Rancho Santa Fe, CA)
Assignee: GRI BIO, INC.
A61K31/7032A61K31/07A61K31/192A61K31/203A61K31/4436A61K45/06Y02A50/30
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Quick Facts
Patent No.
US 11,660,309
App. No.
17/182,098
Granted
May 30, 2023
Kind
B2
Abstract

The present embodiments relate to methods for the prevention and treatment of inflammatory conditions such as alcoholic liver disease (ALD). More specifically the present embodiments relate to the prevention and treatment of ALD through the administration of an Retinoic Acid Receptor (RAR) agonist. Some embodiments relate to use of tazarotene in the prevention and treatment of alcohol-induced liver injury, alcohol-related liver disease, fatty liver disease, hepatic steatosis, alcoholic hepatitis or alcoholic cirrhosis.

Claims (10)

1. A method of inhibiting pro-inflammatory type I NKT cells in a subject, comprising administering an RARγ-selective agonist, wherein the administered RARγ-selective agonist inhibits activation of pro-inflammatory type I NKT cells in the subject.

2. The method of claim 1 , wherein the RARγ-selective agonist is ATRA, retinol, 9-cis-RA, 13-cis-RA, tretinoin, AM580, AC55649, CD1530, or Tazarotene.

3. The method of claim 2 , wherein the RARγ-selective agonist is Tazarotene.

4. The method of claim 1 , wherein the amount of the RARγ-selective agonist is about 1 mg/day to about 10 mg/day.

5. A method of treating an inflammatory condition of fibrosis in a subject in need thereof, the method comprising administering an amount of RARγ-selective agonist sufficient to inhibit activation of pro-inflammatory type I NKT cells to the subject, wherein the fibrosis is associated with an increase in pro-inflammatory type I NKT cells and the administered RARγ-selective agonist inhibits activation of pro-inflammatory type I NKT cells in the subject, thereby treating the inflammatory condition of fibrosis.

6. The method of claim 5 , wherein the administering is by oral delivery.

7. The method of claim 5 , wherein the administering is by pulmonary delivery.

8. The method of claim 5 , wherein the RARγ-selective agonist is ATRA, retinol, 9-cis-RA, 13-cis-RA, tretinoin, AM580, AC55649, CD1530, or Tazarotene.

9. The method of claim 8 , wherein the RARγ-selective agonist is Tazarotene.

10. The method of claim 5 , wherein the amount of the RARγ-selective agonist is about 1 mg/day to about 10 mg/day.

Assignments (3)
SECURITY INTEREST Recorded Dec 15, 2022
From: GRI BIO, INC.
To: ALTIUM GROWTH FUND, LP
Reel/Frame 062108/0599 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 12, 2021
From: CHATURVEDI, VIPIN KUMAR
To: GLYCOREGIMMUNE, INC.
Reel/Frame 055580/0719 →
CHANGE OF NAME Recorded Mar 12, 2021
From: GLYCOREGIMMUNE, INC.
To: GRI BIO, INC.
Reel/Frame 055583/0823 →
Continuity (4)
Continuation 15913541 · Mar 6, 2018
Continuation 14128566
Provisional Application 61501139 · Jun 24, 2011
Related Publication 20210169909A1 · Jun 10, 2021