IP Library Granted Patent US 11,707,485
Granted Patent B2
US 11,707,485 · App. 17/525,577 · Granted Jul 25, 2023

ECM hydrogel for treating esophageal inflammation

Inventors: Stephen Francis Badylak (West Lafayette, IN); Juan Diego Naranjo Gutierrez (Manizales, CO); Lindsey Tamiko Saldin (El Segundo, CA)
Assignee: University of Pittsburgh—Of the Commonwealth System of Higher Education
A61K35/12A61K9/06A61P1/04
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Quick Facts
Patent No.
US 11,707,485
App. No.
17/525,577
Granted
Jul 25, 2023
Kind
B2
Abstract

Methods are disclosed for inhibiting esophageal inflammation in a subject, that include administering to the esophagus of the subject with esophageal inflammation a therapeutically effective amount of an extracellular matrix (ECM) hydrogel. Methods are also disclosed for reducing esophageal stricture. Compositions are disclosed that include an esophageal extracellular matrix (ECM) hydrogel.

Claims (22)

1. A method for inhibiting esophageal inflammation or reducing esophageal stricture in an esophagus of a subject, comprising:

administering to the esophagus of the subject a therapeutically effective amount of an extracellular matrix (ECM) digest solution comprising a hydrated, decellularized, enzymatically digested, extracellular matrix that has not been cross-linked or dialyzed, wherein the digest solution has a pH of about 7.2 to about 7.8 and forms a gel when warmed to a temperature greater than 25° C.,

thereby inhibiting esophageal inflammation or reducing esophageal stricture in the subject.

2. The method of claim 1 , wherein the ECM digest solution is terminally sterilized.

3. The method of claim 1 , wherein the ECM digest solution forms a gel when warmed to about 37° C.

4. The method of claim 1 , wherein the extracellular matrix is derived from urinary bladder, intestine, liver, esophagus, or dermis.

5. The method of claim 1 , wherein the extracellular matrix is from a monkey, horse, pig, cow, or sheep.

6. The method of claim 1 , wherein the digest solution is administered to the subject orally by swallowing or gavage.

7. The method of claim 1 , wherein the digest solution is administered to the esophagus by endoscopy or catheter.

8. The method of claim 1 , wherein the digest solution forms a gel that coats the mucosa of the esophagus upon administration to the subject at about 37° C.

9. The method of claim 1 , wherein the subject has Barret's esophagus.

10. The method of claim 1 , wherein the enzymatically digested ECM is present in the digest solution at a concentration of about 2 mg/mL to about 16 mg/mL.

11. The method of claim 1 , wherein the digest solution is administered at about 37° C.

12. The method of claim 1 , wherein the ECM digest solution is maintained below 37° C. prior to administering to the subject.

13. The method of claim 1 , wherein the ECM digest solution is maintained at or below 25° C. prior to administering to the subject.

14. The method of claim 1 , wherein the subject does not exhibit symptoms of esophageal adenocarcinoma (EAC).

15. The method of claim 1 , wherein the subject does not have, or has not previously had, gastroesophageal reflux disease.

16. The method of claim 1 , wherein the subject has dysplasia of the esophagus.

17. The method of claim 1 , further comprising administering to the subject a therapeutically effective amount of a proton pump inhibitor and/or a histamine antagonist.

18. The method of claim 1 , wherein administering the therapeutically effective amount of the ECM digest solution coats a surface of the lumen of the esophagus.

19. The method of claim 1 , further comprising:

measuring inflammation in the esophagus of the subject.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 15, 2021
From: BADYLAK, STEPHEN FRANCIS; NARANJO GUTIERREZ, JUAN DIEGO; SALDIN, LINDSEY TAMIKO
To: UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION
Reel/Frame 058112/0100 →
Continuity (3)
Continuation 16490054
Provisional Application 62465985 · Mar 2, 2017
Related Publication 20220249549A1 · Aug 11, 2022
Cited By (3)
US 12,383,243 US 12,605,489 US 12,734,274