IP Library › Granted Patent US 12,152,068
Granted Patent B2
US 12,152,068 · App. 17/569,377 · Granted Nov 26, 2024

Binding moieties for biofilm remediation

Inventors: Lawrence M. Kauvar (San Francisco, CA); Stefan Ryser (Menlo Park, CA); Angeles Estelles (Belmont, CA); Reyna J. Simon (Los Gatos, CA); Lauren Opremcak Bakaletz (Columbus, OH); Steven David Goodman (Columbus, OH)
Assignee: Trellis Bioscience, LLC
C07K16/1271A61K39/40A61K45/06A61K49/00C07K14/31C07K16/1214C07K16/1228C07K16/1242C07K16/1275C12Q1/18G01N33/566G01N33/56911A61K35/12A61K39/00A61K2039/505C07K2317/21C07K2317/33C07K2317/34C07K2317/76C07K2317/92C07K2319/00C12N15/86G01N2333/195G01N2333/21G01N2333/245G01N2333/26G01N2333/285G01N2469/10
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Quick Facts
Patent No.
US 12,152,068
App. No.
17/569,377
Granted
Nov 26, 2024
Kind
B2
Abstract

Binding agents able to disrupt bacterial biofilms of diverse origin are described, including monoclonal antibodies secreted by human B lymphocytes. Methods to prevent formation of or to dissolve biofilms with these binding agents are also described. Immunogens for eliciting antibodies to disrupt biofilms are also described.

Claims (25)

1. A monoclonal antibody (mAb) or antigen binding fragment thereof that specifically binds a DNA binding protein II (DNABII), wherein the mAb or antigen binding fragment thereof comprises:

a heavy chain variable region (SEQ ID NO:1) and a light chain variable region (SEQ ID NO: 2) of TRL1068;

a heavy chain variable region (SEQ ID NO:21) and a light chain variable region (SEQ ID NO: 22) of TRL1330; or,

a heavy chain variable region (SEQ ID NO:25) and a light chain variable region (SEQ ID NO: 26) of TRL1337.

2. The mAb or antigen binding fragment thereof of claim 1 , wherein mAb is an Fv antibody, a bispecific antibody, a chimeric antibody, or antigen binding fragment thereof.

3. The mAb or antigen binding fragment thereof of claim 1 , wherein the mAb is a complete antibody.

4. The mAb or antigen binding fragment thereof of claim 3 , wherein the complete antibody comprises generic constant regions heterologous to the variable regions thereof.

5. The mAb or antigen binding fragment thereof of claim 1 , wherein the mAb or antigen binding fragment thereof has an affinity for the DNANH-DNABIL protein that exceeds an affinity of the DNABII protein for a component of a biofilm that includes the DNABII protein.

6. The mAb or antigen binding fragment thereof of claim 1 , wherein the mAb or antigen binding fragment thereof binds a DNABII protein from at least three different bacterial species.

7. The mAb or antigen binding fragment thereof of claim 3 , wherein the mAb or antigen binding fragment thereof (i) has an affinity for the DNABII protein that exceeds an affinity of the DNABII protein for a component of a biofilm that includes the DNABII protein and (ii) binds DNABII protein from at least three different bacterial species.

8. A pharmaceutical or veterinary composition which comprises as an active ingredient the mAb or antigen binding fragment thereof of claim 1 and a suitable pharmaceutical excipient.

9. The pharmaceutical or veterinary composition of claim 8 , further comprising at least one antibiotic and at least one additional active ingredient, the active ingredient comprising an immunostimulant, an antipyrogenic, or an analgesic.

10. A monoclonal antibody (mAb) that specifically binds a DNA binding protein II (DNABII), the antibody comprising:

a heavy chain variable region of (SEQ ID NO:1) and a light chain variable region (SEQ ID NO: 2) of TRL1068;

a heavy chain variable region of (SEQ ID NO:21) and a light chain variable region (SEQ ID NO: 22) of TRL1330; or,

a heavy chain variable region of (SEQ ID NO:25) and a light chain variable region (SEQ ID NO: 26) of TRL1337; and

wherein the mAb is an Fv antibody, a bispecific antibody, a chimeric antibody, or a complete antibody and wherein the complete antibody comprises generic constant regions heterologous to the variable regions thereof.

11. The mAb of claim 10 , wherein the mAb binds a DNABII protein from at least three different bacterial species.

12. A pharmaceutical or veterinary composition which comprises as an active ingredient the mAb of claim 10 and a suitable pharmaceutical excipient.

13. The pharmaceutical or veterinary composition of claim 12 , further comprising at least one antibiotic and at least one additional active ingredient, the active ingredient comprising an immunostimulant, an antipyrogenic, or an analgesic.

14. A monoclonal antibody (mAb) that specifically binds a DNA binding protein II (DNABII), wherein (i) the mAb is an Fv antibody, a bispecific antibody, a chimeric antibody, or a complete antibody, wherein (ii) the mAb comprises a heavy chain variable region of (SEQ ID NO:1) and a light chain variable region (SEQ ID NO: 2) of TRL1068, and wherein (iii) the complete antibody comprises generic constant regions heterologous to the variable regions thereof.

15. The mAb of claim 14 , wherein the mAb binds DNABII protein from at least three different bacterial species.

16. The mAb of claim 14 , wherein the mAb or antigen binding fragment thereof has an affinity for the DNABII protein that exceeds an affinity of the DNABII protein for a component of a biofilm that includes the DNABII protein.

17. A pharmaceutical or veterinary composition which comprises as an active ingredient the mAb of claim 14 and a suitable pharmaceutical excipient.

18. The pharmaceutical or veterinary composition of claim 17 , further comprising at least one antibiotic and at least one additional active ingredient, the active ingredient comprising an immunostimulant, an antipyrogenic, or an analgesic.

Continuity (10)
Continuation 16746708 · Jan 17, 2020
Division 16181260 · Nov 5, 2018
Division 15144681 · May 2, 2016
Continuation In Part 15042061 · Feb 11, 2016
Continuation In Part 14789842 · Jul 1, 2015
Continuation In Part 14668767 · Mar 25, 2015
Continuation In Part 14497147 · Sep 25, 2014
Provisional Application 61926828 · Jan 13, 2014
Provisional Application 61883078 · Sep 26, 2013
Related Publication 20220259294A1 · Aug 18, 2022