Patent Assignment
Reel/Frame 028413/0927
Change of Name
Recorded: 2012-06-20
Pages: 24
Assignor
SANOFI-AVENTIS
Executed: 2011-05-11
Assignee
SANOFI
54 RUE LA BOETIE, PARIS, 75008, FRANCE
Covered Properties
(559)
Dextro-Rotatory Enantiomer of Methyl Alpha-5 (4,5,6,7-Tetrahydro (3,2- C) Thieno Pyridyl) (2-Chlorophenyl)-Acetate and the Pharmaceutical Compositions Containing It
Patent:
4,847,265 →
Application:
07/155,550 →
Alkylaminoalkyl Derivatives of Benzothiophene,Indole and Indolizine, Process for Their Preparationand Compositions Containing Them
Patent:
5,223,510 →
Application:
07/736,580 →
Iontophoresis Device for Transcutaneous Administration of a Given Total Quantity of an Active Principle to a Subject
Patent:
5,320,731 →
Application:
08/016,888 →
Process for the Preparation of a Biphenyl Derivative
Patent:
5,288,895 →
Application:
08/045,519 →
Method for the Secondary Prevention of Ischemic Events
Patent:
5,576,328 →
Application:
08/190,332 →
Method of Promoting Bone Repair Using Tiludronic Disodium Salt
Patent:
5,488,041 →
Application:
08/222,240 →
3-Deoxy Oligosaccharides and Pharmaceutical Compositions Containing Them
Patent:
5,514,659 →
Application:
08/230,921 →
Use of Polyamine Antagonists for the Treatment of Glaucoma
Patent:
5,710,165 →
Application:
08/271,290 →
Method of Treating or Preventing Cardiac Arrhythmia Employing an N-Substituted Heterocyclic Derivative
Patent:
5,541,209 →
Application:
08/293,985 →
Alfuzosin Hydrochloride Dihydrate
Patent:
5,545,738 →
Application:
08/364,180 →
Stable Freeze-Dried Formulation Comprising a Protein Assay Kit
Patent:
5,763,409 →
Application:
08/432,839 →
Method of Preparing a Taxol Derivative
Patent:
6,911,549 →
Application:
08/454,210 →
Oxazoloquinolinone Derivatives, Their Preparation and Their Therapeutic Application as Inhibitors of Monoamine Oxidase
Patent:
5,641,785 →
Application:
08/523,508 →
Process for the Preparation of a Tetrazole Derivative in Two Crystalline Forms and Novel the Crystalline Forms Thereof
Patent:
5,629,331 →
Application:
08/544,027 →
Stable Liquid Composition Containing Urate Oxidase and Lyophilized Composition for Its Preparation
Patent:
5,811,096 →
Application:
08/644,163 →
Iontophoresis Device Comprising at Least One Electrode Assembly with a Reversible Composite Electrode
Patent:
5,807,305 →
Application:
08/776,184 →
Cosmetic Composition Containing a Neuropeptide Y Receptor Antagonist
Patent:
5,827,853 →
Application:
08/790,761 →
Type-2 Neurotensin Receptor (Nt-R2)
Patent:
6,022,856 →
Application:
08/858,876 →
Iontophoresis Device for the Transcutaneous Delivery of an Active Principle Such as an Anionic Oligosaccharide
Patent:
5,928,185 →
Application:
08/875,106 →
Heparin-Like Derivatives
Patent:
5,872,110 →
Application:
08/876,107 →
Use of Fumagillol and Derivatives Thereof for Preparing Medicaments Against Intestinal Infections
Patent:
5,900,431 →
Application:
08/913,360 →
Pharmaceutical Composition for Transdermal Administration
Patent:
6,010,716 →
Application:
08/930,004 →
Oxazolidinone Derivatives, Their Preparation and Therapeutical Use
Patent:
5,843,975 →
Application:
08/973,246 →
Pharmaceutical Amiodarone Composition for Parenteral Delivery
Patent:
6,143,778 →
Application:
08/981,634 →
Quinolein-2(1H)-One Derivatives as Serotonin Antagonists
Patent:
5,958,924 →
Application:
09/011,482 →
Stable Freeze-Dried Pharmaceutical Formulation
Patent:
6,284,277 →
Application:
09/066,387 →
5-Phenyl-3-(Piperidin-4-Yl)-1,3,4-Oxadiazol-2(3H)-One Derivatives for Use as 5-HT4 or H3 Receptor Ligands
Patent:
5,929,089 →
Application:
09/068,390 →
Pyrazole Derivatives, Method for Preparing Same, and Pharmaceutical Compositions Containing Said Derivatives
Patent:
6,028,084 →
Application:
09/068,869 →
3-Pyrazolecarboxamide Derivatives Having Cannabinoid Receptor Affinity
Patent:
5,925,768 →
Application:
09/077,767 →
New Associations of Active Principles Containing Clopidogrel and an Antithrombotic Agent
Patent:
5,989,578 →
Application:
09/117,904 →
Use of Il-7 for Treating Auto-Immune Diseases and Insulin-Dependent Diabetes Mellitus in Particular
Patent:
6,713,053 →
Application:
09/125,168 →
Slow-Release Pharmaceutical Formulations Containing Mizolastine
Patent:
6,165,507 →
Application:
09/125,810 →
Tablet with Controlled Release of Alfuzosine Chlorhydrate
Patent:
6,149,940 →
Application:
09/147,581 →
Process for the Preparation of a Cyanobiphenyl
Patent:
6,392,080 →
Application:
09/147,787 →
Carbohydrate Derivatives
Patent:
6,174,863 →
Application:
09/193,901 →
Synthetic Polysaccharides, Preparation Method Therefor and Pharmaceutical Compositions Containing Same
Patent:
6,534,481 →
Application:
09/230,139 →
Antithrombotic and Antiatherogenic Pharmaceutical Composition Including a Thienopyridine Derivative and an Hmg-Coa-Reductase Inhibitor
Patent:
6,218,403 →
Application:
09/230,299 →
Method for Preparing 4-Methyl-Biphenyl Derivatives
Patent:
6,407,253 →
Application:
09/269,101 →
Device for Ionophoresis Comprising at Least a Membrane Electrode Assembly, for the Transcutaneous Administration of Active Principles to a Subject
Patent:
6,064,908 →
Application:
09/284,971 →
Process for Selective Oxidation of Primary Alcohols of Oligosaccharides
Patent:
6,310,200 →
Application:
09/357,502 →
Method for Preparing 2-Thienylethylamine Derivatives
Patent:
6,080,875 →
Application:
09/380,450 →
Use of Mizolastine for Treating Inflammatory Diseases Associated with 5-Lipoxygenase
Patent:
6,140,335 →
Application:
09/403,005 →
Intermediates and Process for the Preparation Thereof
Patent:
6,215,005 →
Application:
09/423,548 →
Process for the Preparation of a Pharmacologically Active Substance
Patent:
6,180,793 →
Application:
09/423,549 →
Intermediates and Process for the Preparation Thereof
Patent:
6,258,961 →
Application:
09/423,801 →
Use of Oligosaccharide for Preventing Blood Clotting in Extracorporeal Blood Circuits
Patent:
6,391,339 →
Application:
09/424,626 →
Compositions for Treating and Preventing Arterial Thrombosis and Use of a Factor Xa Inhibitor on Its Own and/or Combined with a Platelet Antiaggregating Agent
Patent:
6,541,488 →
Application:
09/445,555 →
Use of a Specific Antagonist of 5HT2 Receptors for Preparaing Medicines Useful for Treating Sleep-Disordered Breathing
Patent:
6,143,792 →
Application:
09/446,484 →
Solid Pharmaceutical Compositions Containing Benzofurane Derivatives
Patent:
7,323,493 →
Application:
09/446,601 →
Process for the Preparation of 1,3-Diaza-Spiro (4.4) Non-1-En-4-One Derivatives and 1-Cyano-1-Acylaminocyclopentane Intermediates
Patent:
6,211,382 →
Application:
09/463,357 →
Process for the Preparation of Imidazolones
Patent:
6,162,923 →
Application:
09/463,433 →
Process for the Preparation of 1,3-Diaza-Spiro (4.4) Non-1-En-4-One Derivatives and 1-Cyano-1-Acylamino-Cyclopentane Intermediates
Patent:
6,239,286 →
Application:
09/463,434 →
4-Oxo-3,5-Dihydro-4H-Pyridazino[4,5-B]-Indole-1-Acetamide Derivatives, Their Preparation and Their Application in Therapy
Patent:
6,262,045 →
Application:
09/463,634 →
Process for the preparation of organic azides
Patent:
6,232,451 →
Application:
09/499,685 →
Hydroxyacetic Ester Derivatives, Preparation Method and Use as Synthesis Intermediates
Patent:
6,573,381 →
Application:
09/509,879 →
Method for Preparing Bromomenthyl-Biphenyl Derivatives
Patent:
6,214,999 →
Application:
09/554,566 →
Synthetic Polysaccharides, Their Method of Production and Pharmaceutical Compositions Containing Same
Patent:
6,528,497 →
Application:
09/600,506 →
Novel Pentasaccharides Processes for Their Preparation and Pharmaceutical Compositions Containing Them
Patent:
6,670,338 →
Application:
09/600,516 →
Device for Automatic Injection of a Dose of Medicinal Product
Patent:
6,575,939 →
Application:
09/601,473 →
Polymorphic Clopidogrel Hydrogenesulphate Form
Patent:
6,429,210 →
Application:
09/623,333 →
Methyl-Phenyl Derivatives, Preparation Method and Use
Patent:
6,417,400 →
Application:
09/646,629 →
Novel Form of Irbesartan, Methods for Obtaining Said Form and Pharmaceutical Compositions Containing Same
Patent:
6,800,761 →
Application:
09/720,017 →
Disposable Injection Device Designed to Be Pre-Filled
Patent:
6,432,090 →
Application:
09/806,569 →
Disposable Injection Device Designed to Be Pre-Filled
Patent:
6,447,480 →
Application:
09/806,574 →
Pharmaceutical Composition with Gastric Residence and Controlled Release
Patent:
6,861,072 →
Application:
09/807,573 →
Process for Racemization
Patent:
6,670,486 →
Application:
09/830,930 →
1,4-Diazabicylo[3,2,2] Nonane Derivatives, Their Preparation and Their Therapeutic Application
Patent:
6,407,095 →
Application:
09/856,945 →
Controlled-Release Dosage Forms Comprising Zolpidem or a Salt Thereof
Patent:
6,514,531 →
Application:
09/857,154 →
Pyrazolecarboxylic Acid Derivatives, Their Preparation, Pharmaceutical Compositions Containing Them
Patent:
6,432,984 →
Application:
09/890,242 →
Stable Formulation Containing Fumagillin
Patent:
6,528,539 →
Application:
09/913,547 →
Pyridopyranoazepine Derivatives, Their Preparation and Their Therapeutic Application
Patent:
6,538,003 →
Application:
09/913,679 →
1,4-Diazabicyclo[3.2.2]Nonane-4-Carboxylates and Carboxamide Derivates, Production and Use Thereof in Therapeutics
Patent:
6,987,106 →
Application:
09/937,045 →
Novel Morpholine Derivatives, Method for the Production Thereof and Pharmaceutical Preparations Containing Said Derivatives
Patent:
6,506,750 →
Application:
09/937,279 →
Process for the Preparation of Fumagillin
Patent:
6,521,764 →
Application:
10/009,116 →
Disposable Injection Device
Patent:
6,918,889 →
Application:
10/009,264 →
Aminothiazole Derivatives and Their Use as Crf Receptor Ligands
Patent:
6,586,456 →
Application:
10/031,038 →
Phenyl-And Pyridyl-Tetrahydro-Pyridines Having Tnf Inhibiting Activity
Patent:
6,509,351 →
Application:
10/111,045 →
Method for Preparing a Thiopene Derivative
Patent:
6,639,083 →
Application:
10/111,159 →
Pyrazolecarboxylic Acid Tricyclic Derivatives, Preparation and Pharmaceutical Compositions Containing Same
Patent:
6,906,080 →
Application:
10/111,765 →
Safety System for a Syringe
Novel Branched Substituted Amino Derivatives of 3-Amino-1-Phenyl-1H-[1,2,4] Triazol, Methods for Producing Them and Pharmaceutical Compositions Containing Them
Pyrazolecarboxylic Acid Derivatives, Their Preparation and Pharmaceutical Compositions Containing Them, and Method of Treating
4-Heteroparyl-1,4-Diazabicyclo[3.2.2]Nonane, Preparation and Therapeutic Use Thereof
Novel 1,3-Dihydro-2H-Indol-2-One Derivatives and Their Use as Ligands for V1B and V1A Arginine-Vasopressin Receptors
2-Amino-3-(Alkyl)-Pyrimidone Derivatives as GSK3.Beta. Inhibitors
1,4-Diazabicyclo[3.2.2]Nonabenzoxazole, -Benzothiazole and Benzimidazole Derivatives, Preparation and Therapeutic Use Thereof
1,4-Diazabicyclo[3.2.2]Nonane-Phenylisoxazole Derivatives, Their Preparation and Their Application in Therapeutics
4-(2 Phenylthiazol-5-Yl)-1, 4-Diazabicyclo-[3.2.2]Nonane Deirvatives, Preparation and Therapeutic Use Thereof
Device for Protecting a Syringe Needle
Pyridopyranoazepine Derivatives, Their Preparation and Their Therapeutic Application
Aminoalkoxybenzoyl-Benzofuran or Benzothiophene Derivatives, Method for Preparing Same and Compositions Containing Same
Aminoalkenylbenzoyl-Benzofuran or Benzothiophene, Method for Preparing Same and Compositions Containing Same
Aminoalkoxybenzoyl-Benzofuran or Benzothiophene Derivatives, Method of Preparing Same and Compositions Containing Same
2-Pyridinyl-6,7,8,9-Tetrahydropyrimido{1,2-A}Pyrimidin-4-One and 7-Pyridinyl-2,3-Dihydoimidazo{1,2-a}Pyrimidin-5(1H)One Derivatives
1-[Alkyl],1-[(Heteroaryl)Alkyl] and 1-[Aryl]Alkyl]-7PYRIDINYL-Imidazo[1,2-Alpha]Pyrimidin-5(1H)-One Derivatives
Polysaccharides with Antithrombotic Activity Comprising at Least a Covalent Bond with Biotin or a Biotin Derivative
Hydroxyacetic Ester Derivatives, Preparation Method and Use as Synthesis Intermediates
Cyclohexyl(Alkyl)-Propanolamines, Preparation Method and Pharmaceutical Compositions Containing Same
2-Butyl-3-(4-[3(Dibutylamino)Propoxy]Benzoyl)-5-Nitro-Benzofuran Hydrochloride and Preparation Thereof
Methanesulphonamido-Benzofuran, Preparation Method and Use Thereof as Synthesis Intermediate
Pharmaceutical Dronedarone Composition for Parenteral Administration
Derivatives of N-(Arylsulfonyl)Beta-Aminoacids Comprising a Substituted Aminomethyl Group, the Preparation Method Thereof and the Pharmaceutical Compositions Containing Same
Pharmaceutical Combinations Based on Pyridoindolone Derivatives and Anticancer Agents
Use of Pyridoindolone Derivatives for Preparing Anticancer Medicines
Chloromethylation of Thiophene
Aminoquinoline and Aminopyridine Derivatives and Their Use as Adenosine A3 Ligands
Acylaminothiazole Derivatives, Their Preparation and Therapeutic Use
3-Substituted-4-Pyrimidone Derivatives
Substituted 2-Pyridinyl-6,7,8,9-Tetrahydropyrimido{1,2-a}Pyrimidin-4-One and 7-Pyridinyl-2,3-Dihydroimidazo{1,2-a}Pyrimidin-5(1H)One Derivatives
Substituted 2-Pyrimidinyl-6,7,8,9-Tetrahydropyrimido[1,2-a]Pyrimidin-4-One and 7-Pyrimidinyl-2,3-Dihydroimidazo[1,2-a]Pyrimidin-5(1H)One Derivatives for Neurodegenerative Disorders
4-(Oxadiazol-3-Yl)-1,4-Diazabicyclo[3.2.2]-Nonane Derivatives, Preparation and Therapeutic Use Thereof
4-(1,3,4,-Thiadiazol-2-Yl)-1,4-Diazabicyclo-[3.2.2]Nonane Derivatives, Preparation and Therapeutic Use Thereof
4-(Oxazolopyridin-2-Yl)-1,4-Diazabicyclo-[3.2.2]Nonane Derivatives, Preparation and Therapeutic Use Thereof
3-Heteroaryl-3, 5-Dihydro-4-Oxo-4H-Pyridazino[4, 5-B]Indole-1-Carboxamide Derivatives Their Preparations and Therapeutic Use
Derivatives of 5-(Pyridin-3-Yl)-1-Azabicyclo[3.2.1] Octane, the Preparation Thereof and the Application of Same in Therapeutics
Idraparinux(SANORG34006)For Treatment of Venous Events in Patients with Deep Venous Thrombosis
Needle Sheathing Device with Flexible End-Piece for Syringe
Heteroaryl Substituted 2-Pyridinyl and 2-Pyrimidinyl-6,7,8,9-Tetrahydropyrimido[1,2-a]Pyrimidin-4-One Derivatives
7-(Pyrimidin-4-Yl)- Imadazo [1,2-a] Pyrimidin-5(1H)-Ones as GSK3BETA Inhibitors
3-Heteroarly-3,5-Dihydro-4-Oxo-4H-Pyridazino[4,5-B] Indole-1-Acetamide Derivatives, Preparation and Use Thereof in Medicaments
Novel 1,2,3-Substituted Indolizine Derivatives, Inhibitors of Fgfs, Method for Making Same and Pharmaceutical Compositions Containing Same
Piperazinylacylpiperidine Derivatives, Their Preparation and Therapeutic Use Thereof
Piperazinylacylpiperidine Derivatives, Their Preparation and Therapeutic Use Thereof
Rigid Plastic Protective Case for a Blister Pack
3-Substituted-4-Pyrimidone Derivatives
2,3,6-Trisubstituted-4-Pyrimidone Derivatives
Use of Antagonists of the Cbi Receptor for the Manufacture of a Composition Useful for the Treatment of Hepatic Diseases
Synthetic Polysaccharides, Process for Their Preparation and Pharmaceutical Compositions Containing Them
Process for Racemization
Hydroxyacetic Ester Derivatives, Preparation Method and Use as Synthesis Intermediates
Novel Form of Irbesartan, Processes for Obtaining the Said and Pharmaceutical Compositions Containing It
2-Amino-3-(Alkyl)-Pyrimidone Derivatives
Novel Polysaccharides with Antithrombotic Activity Comprising at Least One Covalent Bond with Biotin or a Biotin Derivative
Derivatives of Dioxane-2-Alkyl Carbamates, Preparation Thereof and Application Thereof in Therapeutics
1,4-Diazabicyclo[3.2.2]Nonanecarboxamide Derivatives, Preparation and Therapeutic Use Thereof
Pyridoindolone Derivatives Substituted in the 3-Position by a Phenyl, Their Preparation and Their Application in Therapeutics
Pyrazolecarboxylic Acid Tricyclic Derivatives, Preparation and Pharmaceutical Compositions Containing Same
Purified Polypeptides Having Il-13 Receptor Activity
Use of Pyridoindolone Derivatives for the Preparation of Medicinal Products
Substituted 2-(Diaza-Bicyclo-Alkyl)-Pyrimidone Derivatives
Substituted 8'-Pyridinyl-Dihydrospiro-[Cycloalkyl]-Pyrimido[1,2-a]Pyrimidin-6-One and 8'-Pyrimidinyl-Dihydrospiro-[Cycloalkyl]-Pyrimido[1,2-a]Pyrimidin-6-One Derivatives
Process for the Preparation of Pyridinyl and Pyrimidinyl Mono-Fluorinated Beta Keto-Esters
Substituted 8-Perfluoroalkyl-6,7,8,9-Tetrahydropyrimido[1,2-a] Pyrimidin-4-One Derivatives
8-Substituted-6,7,8,9-Tetrahydropyrimido [1,2-a] Pyrimidin-4-One Derivatives
4-Cyanopyrazole-3-Carboxamide Derivatives, Preparation, and Application Thereof
1-[Alkyl], 1-[(Heteroaryl) Alkyl] and 1-[(Aryl)Alkyl]-7-Pyridinyl-Imidazo[1,2-a]Pyrimidin-5(1H)-One Derivatives
Substituted Indolizine 1,2,3,6,7,8 Derivatives, Fgfs Inhibitors, a Method for the Preparation Thereof and Pharmaceutical Compositions Containing Said Derivatives
Derivatives of N-Heterocyclylmethylbenzamides, Prepartion Method Thereof and Application of Same in Therapeutics
4-Phenylpiperazin-1-Yl)Acylpiperidine Derivatives, Preparation Thereof and Application of Same in Therapeutics
Substituted 8'-Pyri(Mi)Dinyl-Dihydrospiro-[Cycloalkylamine]-Pyrimido[1,2-a]Pyrimidin-6-One Derivatives
Pyrazole Derivatives and Use Thereof as Orexin Receptor Antagonists
3-Heteroaryl-3,5-Dihydro-4-Oxo-4H-Pyridazino[4,5-B]Indole-1-Carboxamide Derivatives, Their Preparation and Therapeutic Use
Derivatives of N-' (1,5-Diphenyl-1H-Pyrazol-3-Yl) Sulfonamide with CB1 Receptor Affinity
Dual Molecules Containing Peroxy Derivative, the Synthesis and Therapeutic Applications Thereof
Derivatives of 1,4-Diazabicyclo[3.2.1]Octanecarboxamide, Preparation Method Thereof and Use of Same in Therapeutics
Aryloxyalkylcarbamate-Type Derivatives, Preparation Method Thereof and Use of Same in Therapeutics
Derivatives of N-[(1,5-Diphenyl-1H-Pyrazol-3-Yl)Methyl] Sulfonamide, Their Preparation and Their Application in Therapeutics
Patent:
7,297,710 →
Application:
11/457,014 →
Pyrimidine Derivatives as Orexin Receptor Antagonists
Use of Oligosaccharide for Preventing Blood Clotting in Extracorporeal Blood Circuits
Application:
11/464,259 →
Publication:
US 2007/0197637
Cyclohexyl(Alkyl)Propanolamines, Preparation Method and Pharmaceutical Compositions Containing Same
Antithrombotic Compound
Derivatives of 1-Piperazine-and 1-Homopiperazine-Carboxylates, Preparation Method Thereof and Use of Same as Inhibitors of the Faah Enzyme
1-Amino-Phthalazine Derivatives, the Preparation and the Therapeutic Use Thereof
2H-Or 3H-Benzo[E]Indazol-1-Yl Carbamate Derivatives, the Preparation and Therapeutic Use Thereof
Tetrahydroisoquinoline Sulfonamide Derivatives, the Preparation Thereof, and the Use of the Same in Therapeutics
2-Morpholino-4-Pyrimidone Compound
6- (Pyridinyl) -4-Pyrimidone Derivates as Tau Protein Kinase 1 Inhibitors
4-Arylmorpholin-3-One Derivatives, Their Preparation and Therapeutic Use Thereof
N-(1H-Indolyl)-1H-Indole-2-Carboxamide Derivatives, Their Preparation and Their Therapeutic Use
Laser Radiation Desorption Device for Manipulating a Liquid Sample in the Form of Individual Drops, Thereby Making It Possible to Carry Out the Chemical and Biological Treatment Thereof
Pyrido-Pyrimidine Derivatives, Preparation Thereof, and Therapeutic Use Thereof
Pharmaceutical Composition in the Form of a Gastric-Resident Tablet Containing an Active Principle
Application:
11/675,712 →
Publication:
US 2007/0190140
Pharmaceutical Composition Comprising a Solid Dispersion with a Polymer Matrix Containing a Continuous Polydextrose Phase and a Continuous Phase of a Polymer Other Than Polydextrose
Indolin-2-One Pyridine Derivatives, Preparation and Therapeutic Use Thereof
Method and Intermediates for the Preparation of Derivatives of N (1-Benzhydrylazetidin-3-Yl)-N-Phenylmethylsulfonamide
Use of Substituted 2-(Diaza-Bicyclo-Alkyl)-Pyrimidone Derivatives for the Treatment of Neurodegenerative Diseases
Use of Substituted 8-Perfluoroalkyl-6,7,8,9-Tetrahydropyrimido[1,2-a] Pyrimidin-4-One Derivatives as Therapeutic Agents
Use of Substituted 2-Pyridinyl-6,7,8,9-Tetrahydropyrimido[1,2-a] Pyrimidin-4-One and 7-Pyridinyl-2,3-Dihydroimidazo[1,2-a] Pyrimidin-5(1H)One Derivatives as Therapeutic Agents
Derivatives of 5-(Pyridin-3-Yl)-1-Azabicyclo[3.2.1]Octane, Their Preparation and Their Therapeutic Application
Aminothiazole Derivatives and Their Use as Crf Receptor Ligands
3-Heteroaryl-3,5-Dihydro-4-Oxo-4H-Pyridazino[4,5 B]Indole-1-Acetamide Derivatives, Their Preparation and Their Application in Therapeutics
Heteroaryl Substituted 2-Pyridinyl and 2-Pyrimidinyl -6,7,8,9-Tetrahydropyrimido[1,2-a] Pyrimidin-4-One Derivatives
Use of 8-Substituted-6,7,8,9-Tetrahydropyrimido[1,2-a] Pyrimidin-4-One Derivatives
N-(Heteroaryl)-1H-Indole-2-Carboxamide Derivatives and Their Use as Vanilloid TRPV1 Receptor Ligands
Sulfonyl Pyrrolidines, Method for Producing the Same and Their Use as Drugs
Substituted N-Aminomethylene Sulfonamides, Production and Use Thereof as Medicaments
Substituted 4-Phenyltetrahydroisoquinolines, Pharmaceuitcal Compositions Comprising Them and Therapeutic Methods for Their Use
Tetrahydrofuran Derivatives for Use as Inhibitors of Matrix Metalloproteinases
4-Cyanopyrazole-3-Carboxamide Derivatives, Preparation and Application Thereof
2-Pyridinyl-6,7,8,9-Tetrahydropyrimido[1,2-A] Pyrimidin-4-One and 7-Pyridinyl-2,3-Dihydroimidazo[1,2-a] Pyrimidin-5(1H)One Derivatives
Amide-Substituted 8 N Benzimidazoles, Method for the Production Thereof, and Use of the Same as Medicaments
Substituted 2-Aminoalkylthiobenzimidazole Compounds, Pharmaceutical Compositions Thereof and Methods for Their Use
Substituted, Bicyclic 8-Pyrrolidinobenzimidazoles, Methods for Their Production and Their Use as Medicaments
Aminocarbonyl-Substituted 8-N-Benzimidazoles, Methods for Their Preparation and Their Use in Pharmaceutical Compositions
Amino-Substituted 8-N-Benzimidazoles and Methods for Their Use in Blood Sugar Disorders
Novel Imidazo[1,5-a] Pyridine Derivatives, Method for Preparing Same and Pharmaceutical Compositions Containing Same
Derivatives of N-Heterocyclylmethylbenzamides, Preparation Method Thereof and Application of Same in Therapeutics
Derivatives of N-[(1,5-Diphenyl-1H-Pyrazol-3-Yl)Methyl] Sulfonamide, Their Preparation and Their Application in Therapeutics
Substituted Tetrahydroisochinolines as Mmp Inhibitors, Related Production Method and Use as Medicine
Substituted 8'-Pyridinyl-Dihydrospiro-[Cycloalkyl]-Pyrimido[1,2-a] Pyrimidin-6-One and 8'-Pyrimidinyl-Dihydrospiro-[Cycloalkyl]-Pyrimido[1,2-a] Pyrimidin-6-One Derivatives
Substituted 8'-Pyri(Mi)Dinyl-Dihydrospiro-[Cycloalkylamine]-Pyrimido[1,2-a]Pyrimidin-6-One Derivatives
3-Heteroaryl-3,5-Dihydro-4-Oxo-4H-Pyridazino[4,5-B]Indole-1-Acetamide Derivatives, Their Preparation and Their Application in Therapeutics
Azole Derivatives in the Form of Lipase and Phospholipase Inhibitors
Association Between Ferroquine and an Artemisinine Derivative for Treating Malaria
Application:
11/874,377 →
Publication:
US 2012/0258945
Use of Mgc4504
Application:
11/908,065 →
Publication:
US 2008/0249011
Use of a Gip Promoter Polymorphism
Heteroaryl-Carboxylic Acid (Sulfamoyl Alkyl) Amide - Derivatives as Factor Xa Inhibitors
Method for Producing 2-(2-Aminopyrimidin-4-Yl)-1H-Indole-5-Carboxylic Acid Derivatives
6-Oxazol-4-Ylmetholmethoxy-Alko-Alkoxymethyl Substituted Benzoic Acid Derivatives Forming Peroxisome Proliferator - Activated Receptor (Ppar) Ligands, Process for Their Preparation and Methods of Use Thereof
Hydrates of Alkaline-Earth Salts of Irbesartan and the Preparation Thereof
Azolopyridin-2-One Derivatives as Lipase and Phospholipase Inhibitors
Benzothiazol-2-One Derivatives as Lipase and Phospholipase Inhibitors
Benzooxazol-2-One Derivatives as Lipase and Phospholipase Inhibitors
Derivatives of 4,5-Diarylpyrrole, Preparation Method Thereof and Use of Same in Therapeutics
Substituted Heterocycles, Their Use as Medicament, and Pharmaceutical Preparations Comprising Them
Substituted Heterocycles, Their Use as Medicament, and Pharmaceutical Preparations Comprising Them
Derivatives of Pyrido[2,3-D]Pyrimidine, the Preparation Thereof, and the Therapeutic Application of the Same
Heteroaryl-Substituted Amides Comprising A Saturated Linker Group, And Their Use As Pharmaceuticals
Heteroaryl-Substituted Amides Comprising An Unsaturated Or Cyclic Linker Group, And Their Use As Pharmaceuticals
Isoquinoline Derivatives
Pyrazolopyridine Derivatives as Inhibitors of Beta-Adrenergic Receptor Kinase 1
N-(Heteroaryl)-1-Heteroarylalkyl-1H-Indole-2-Carboxamide Derivatives, Preparation and Therapeutic Use Thereof
N-(Arylalkyl)-1H-Pyrrolopyridine-2-Carboxamide Derivatives, Preparation and Therapeutic Use Thereof
Intermediate Compound for Synthesizing Pharmaceutical Agent and Production Method Thereof
Cyclohexylamin Isoquinolone Derivatives
Piperidinyl-Substituted Isoquinolone Derivatives
Derivatives of 5-Pyridinyl-1-Azabicyclo[3.2.1]Octane, Preparation Method Thereof and Use of Same in Therapeutics
Derivatives of 5-Pyridazinyl-1-Azabicyclo[3.2.1]Octane, Preparation Method Thereof and Use of Same in Therapeutics
Combination of a Long-Acting Hypnotic Agent and a Short-Acting Hypnotic Agent and Therapeutic Use Thereof
Application:
12/029,011 →
Publication:
US 2008/0181943
Substituted 4-Phenyltetrahydroisoquinolines, Process for Their Preparation, Pharmaceutical Compositions and Therapeutic Use
Process for Preparing N-Alkylnaltrexone Halides
Phenyl-[1,2,4]-Oxadiazol-5-One Derivatives, Pharmaceutical Compositions and Therapeutic Use Thereof
Derivatives of 2-Aminothiazoles and 2-Amino-Oxazoles, Processes for Their Preparation and Their Use as Pharmaceutical Compositions
Phenyl-1,2,4-Oxadiazolone Derivatives, Processes for Their Preparation and Methods for Their Use as Pharmaceuticals
Cyclic N-[1,3,4]-Thiadiazol-2-Yl-Benzene Sulfonamides, Pharmaceutical Compositions and Methods for the Therapeutic Use Thereof
Bicyclic Aryl-Sulfonic Acid [1,3,4]-Thiadiazol-2-Yl-Amides, Processes for Their Preparation, Pharmaceutical Compositions and Methods for Their Use
N-[1,3,4]-Thiadiazol-2-Yl-Benzene Sulfonamides, Pharmaceutical Compositions Thereof and Methods for Their Therapeutic Use
4-Oxy-N-[1,3,4]-Thiadiazol-2-Yl-Benzene Sulfonamides, Pharmaceutical Compositions and Methods for Their Therapeutic Use
Bushing for Receiving a Dropper Neck, and Corresponding Package and Kit
Application:
12/085,634 →
Publication:
US 2010/0016826
EGLN2 Variants and Use Thereof in Preventing or Treating Thromboembolic Disorders and Coronary Heart Disease
Diacyl Indazole Derivatives as Lipase and Phospholipase Inhibitors
Triazolopyridine Derivatives as Inhibitors of Lipases and Phospholipases
Carbamoylbenzotriazole Derivatives as Inhibitors of Lipases and Phospholipases
Imidazole Derivatives as Inhibitors of Tafia
Therapeutic Use of N-(1H-Indolyl)-1H-Indole-2-Carboxamide Derivatives
Novel Indolizine Derivatives, Method for Preparing Same, and Therapeutic Compositions Comprising Same
Pyridoindolone Derivatives Substituted in the 3-Position by a Phenyl, Their Preparation and Their Application in Therapeutics
Use of Substituted 2-Pyrimidinyl-6,7,8,9-Tetrahydropyrimido[1,2-a] Pyrimidin-4-One and 7-Pyrimidinyl-2,3-Dihydroimidazo[1,2-a] Pyrimidin-5(1H)One Derivatives
3-Acylindole Derivatives, Preparation and Therapeutic Use Thereof
Substituted Bicyclic Pyrimidone Derivatives
Isoquinoline and Benzo[H]Isoquinoline Derivatives, Preparation and Therapeutic Use Thereof as Antagonists of the Histamine H3 Receptor
N-(Heteroaryl)-1H-Indole-2-Carboxamide Derivatives and Their Use as Vanilloid TRPV1 Receptor Ligands
Cyclohexyl(Alkyl)Propanolamines, Preparation Method and Pharmaceutical Compositions Containing Same
Method for the Determination of the Activity of the Organic Cation Transporter
Application:
12/162,833 →
Publication:
US 2009/0184006
Fgf-Receptor Agonist Dimeric Compounds
Cytotoxic Agents Comprising New Tomaymycin Derivatives
Tricyclic N-Heteroaryl-Carboxamide Derivatives Containing a Benzimidazole Unit, Method for Preparing Same and Their Therapeutic Use
Azacyclyl-Substituted Arylthienopyrimidinones, Process for Their Preparation and Their Use as Medicaments
Novel Azacyclyl-Substituted Aryldihydroisoquinolinones, Process for Their Preparation and Their Use as Medicaments
Amino Alcohol-Substituted Arylthienopyrimidinones, Process for Their Preparation and Their Use as Medicaments
Novel Aminoalcohol-Substituted Aryldihydroisoquinolinones, Process for Their Preparation and Their Use as Medicaments
Method and Intermediates for the Preparation of Derivatives of N (1-Benzhydrylazetidin-3-Yl)-N-Phenylmethylsulfonamide
USE OF 7-(PYRIMIDIN-4 YL)-IMIDAZO[1,2-a]PYRIMIDIN-5(1H)-ONES AS GSK-3BETA INHIBITORS
Application:
12/194,899 →
Publication:
US 2008/0318980
Aryloxyalkylcarbamate-Type Derivatives, Preparation Method Thereof and Use of Same in Therapeutics
Novel 1,2,3-Substituted Indolizine Derivatives, Inhibitors of Fgfs, Method for Preparing Them and Pharmaceutical Compositions Containing Them
Use of Fgf Inhibiting Substituted 1,2,3 Indolizine Derivatives in the Preparation of Medicaments Which Can Be Used to Treat Diseases Linked to Pathological Choroidal Angiogenesis
Use of Idraparinux for Extended Prophylaxis of Thromboembolism
Application:
12/206,095 →
Publication:
US 2010/0062997
Novel Substituted 2-Amino-4-Phenyldihydroquinolines, Processes for Their Preparation, Pharmaceutical Compositions and Methods for Their Use
Substituted 1-Amino-4-Phenyl-Dihydroisoquinolines, Methods for the Production Thereof, Use Thereof as a Medicament, and Medicaments Containing Them
Azolopyridin-3-One Derivatives as Inhibitors of Lipases and Phospholipases
Imidazopyridin-2-One Derivatives as Inhibitors of Lipases and Phospholipases
Dimers of Artemisinin Derivatives, Preparation Thereof and Therapeutic Use Thereof
1,4-Diazabicyclo[3.2.2]nonanecarboxamide Derivatives, Preparation and Therapeutic Use Thereof
Slimming Cosmetic Composition Containing a Substance Inducing the Production of Il-6
Phenylamino-Benzoxazole Substituted Carboxylic Acids, Method for Their Production and Use Thereof as Medicaments
Application:
12/267,896 →
Publication:
US 2009/0149519
4,5-Diphenyl-Pyrimidinyl Substituted Carboxylic Acids, Method for the Production and Use Thereof as Medicaments
4,5-Diphenyl-Pyrimidinylamino Substituted Carboxylic Acids, Method for the Production and Use Thereof as Medicaments
4,5-Diphenyl-Pyrimidinyl-Oxy or -Mercapto Substituted Carboxylic Acids, Method for the Production and Use Thereof as Medicaments
Leptomycin Derivatives
Spirocyclic Nitriles as Protease Inhibitors
2-(Cyclic Amino)-Pyrimidone Derivatives
Use of ADAMTS4 Gene and Protein Polymorphisms
Application:
12/300,200 →
Publication:
US 2010/0062431
Derivatives of 5-Pyridazinyl-1-Azabicyclo[3.2.1]Octane, Preparation Method Thereof and Use of Same in Therapeutics
Urea Derivatives of Tropane, Their Preparation and Their Therapeutic Application
Aryl- and Heteroaryl-Ethyl-Acylguanidine Derivatives, Their Preparation and Their Application in Therapeutics
Derivatives of Imidazo[1,2-a]Pyridine-2-Carboxamides, Preparation Method Thereof and Use of Same in Therapeutics
CXCR2 Inhibitors
Inhibitors of CXCR2
Substituted Quinoxalines, Their Preparation and Their Therapeutical Use as 11BETAHSD1 Modulators
CXCR2 Antagonists
CXCR2 Inhibitors
Regioselective Palladium Catalyzed Synthesis of Benzimidazoles and Azabenzimidazoles
Antitumor Combinations Containing Taxane Derivatives
Application:
12/356,668 →
Publication:
US 2009/0196869
Pyrazolo[4,3-D]Thiazole Derivatives, and Preparation and Therapeutic Application Thereof
N-(Aminoheteroaryl)-1H-Indole-2-Carboxamide Derivatives, Preparation Thereof and Therapeutic Use Thereof
N-(Aminoheteroaryl)-1H-Indole-2-Carboxamide Derivatives, and Preparation and Therapeutic Application Thereof
Derivatives of Pyrido[2,3-D]Pyrimidine, the Preparation Thereof, and the Therapeutic Application of the Same
Imino-Imidazo-Pyridine Derivatives Having Antithrombotic Activity
Arylaminoaryl-Alkyl-Substituted Imidazolidine-2,4-Diones, Process for Preparing Them, Medicaments Comprising These Compounds, and Their Use
Use of Cyclipostin Derivatives for the Treatment of Mycobacterial Infectious Diseases
5,6-Bisaryl-2-Pyridine-Carboxamide Derivatives, Preparation and Application Thereof in Therapeutics as Urotensin Ii Receptor Antagonists
EPHA2 Receptor Antagonist Antibodies
Tartrate Derivatives for Use as Coagulation Factor Ixa Inhibitors
Isoserine Derivatives for Use as Coagulation Factor Ixa Inhibitors
2-Aryl-6-Phenylimidazo[1,2-A]Pyridine Derivatives, Preparation Thereof and Therapeutic Use Thereof
Substituted 2-Phenyl-Benzimidazoles and Their Use as Pharmaceuticals
Pyrido-Pyrimidine Derivatives, Preparation Thereof, and Therapeutic Use Thereof
New Imidazolone Derivatives, Preparation Thereof as Drugs, Pharmaceutical Compositions, and Use Thereof as Protein Kinase Inhibitors, in Particular CDC7
Isolated Peptides from Actinomadura Namibiensis
Use of Dronedarone for the Preparation of a Medicament for Use in the Prevention of Cardiovascular Hospitalization or of Mortality
Use of Dronedarone for the Treatment of Patients with Arrhythmia and Having an Increase of Creatinine Level Due to Dronedarone Administration
Application:
12/431,830 →
Publication:
US 2010/0016423
SUBSTITUTED 8-PIPERIDINYL-2-PYRIDINYL-PYRIMIDO[1,2-a] PYRIMIDIN-6-ONE AND 8-PIPERIDINYL-2-PYRIMIDINYL-PYRIMIDO[1,2-a] PYRIMIDIN-6-ONE DERIVATIVES
Application:
12/434,053 →
Publication:
US 2009/0281121
Substituted Pyrazoles, Compositions Containing These, Method of Production and Use
Novel Anti-CD38 Antibodies for the Treatment of Cancer
Nicotinic Acetylcholine Receptor Sub-Type Selective Amides of Diazabicycloalkanes
Pyrrole Derivatives, Preparation Thereof and Therapeutic Use Thereof
Imidazo[2,1-B]Thiazoles and Their Use as Pharmaceuticals
Phenyl-1,2,4-Oxadiazolone Derivatives with Phenyl Group, Processes for Their Preparation and Their Use as Pharmaceuticals
Use of Irbesartan for the Preparation of Medicinal Products That Are Useful for Treating Pulmonary Hypertension
Urea and Sulfamide Derivatives as Inhibitors of Tafia
Sulfonyl-Phenyl-2H-[1,2,4]Oxadiazol-5-One Derivatives , Processes for Their Preparation and Their Use as Pharmaceuticals
Method for the Diastereoselective Production of a Chiral Primary Amine on a Steroid
Application:
12/483,365 →
Publication:
US 2010/0069627
5-Alkyloxy-Indolin-2-One Derivatives, Preparation Thereof and Application Thereof in Therapy
Application:
12/483,782 →
Publication:
US 2010/0069384
Novel Therapeutic Use for Treating of Leukemia
Heteroarylacrylamides and Their Use as Pharmaceuticals
Heteroarylcyclopropanecarboxamides and Their Use as Pharmaceuticals
Heteroaryl-Substituted Carboxamides and Their Use as Pharmaceuticals
Substituted Heteroaryl Pyridopyrimidone Derivatives
Cycloalkylamine substituted isoquinoline derivatives
Substituted Isoquinoline and Isoquinolinone Derivatives as Inhibitors of Rho-Kinase
New substituted isoquinoline and isoquinolinone derivatives
Substituted isoquinoline and isoquinolinone derivatives
Cycloalkylamine Substituted Isoquinolone Derivatives
Cycloalkylamine Substituted Isoquinoline and Isoquinolinone Derivatives
Cycloalkylamine substituted isoquinolone and isoquinolinone derivatives
Application:
12/487,525 →
Publication:
US 2010/0056568
3-Heteroaryl-3,5-Dihydro-4-Oxo-4H-Pyridazino[4,5-B]Indole-1-Carboxamide Derivatives, Their Preparation and Therapeutic Use
Application:
12/487,902 →
Publication:
US 2009/0275576
N-(Amino-Heteroaryl)-1H-Pyrrolopyridine-2-Carboxamides Derivatives Preparation Thereof and Their Use in Therapy
Use of Substituted Pyranone Acid Derivatives for the Treatment of Metabolic Syndrome
Derivatives of Pyrrolopyridine-2-Carboxamides, Preparation Thereof and Therapeutic Application Thereof
Derivatives of N-(Heteroaryl)-1-Heteroaryl-1H-Indole-2-Carboxamides, Preparation Thereof and Therapeutic Use Thereof
Therapeutic Use of N-(1H-Indolyl)-1H-Indole-2-Carboxamide Derivatives
Phenothiazin Derivates, Method for the Production Thereof and Use Thereof as Pharmaceuticals
Derivatives of Dioxan-2-Alkyl Carbamates, Preparation Thereof and Application Thereof in Therapeutics
2-Substituted-6-Heterocyclic Pyrimidone Derivatives as Tau Protein Kinase 1 Inhibitors
Bio-Active Peptide Hormone
Application:
12/519,978 →
Publication:
US 2010/0184660
Blister Protection Sleeve Including Automatic Locking Means That Can Be Unlocked by Torsion
Fluorescence-Based Assay for Detecting Compounds for Modulating the Sodium-Calcium Exchanger (Ncx) in "Forward Mode"
Application:
12/529,230 →
Publication:
US 2010/0151497
Method for Producing Peptide Libraries and Use Thereof
Application:
12/529,780 →
Publication:
US 2010/0234246
Azabicycloalkane Derivatives, Preparation Thereof and Use Thereof in Therapy
Use of a Compound Antagonist to the NK2 Receptors of Neurokinin a for the Preparation of Drugs Useful for Preventing and Treating of Sexual Dysfunction
Application:
12/537,345 →
Publication:
US 2010/0173879
Low Molecular Weight Heparins Including at Least One Covalent Bond with Biotin or a Biotin Derivative, Method for Making Same and Use Thereof
Application:
12/539,224 →
Publication:
US 2010/0081629
Amorphous Solid Composition Containing a Pyrazole-3-Carboxamide in Amorphous Form and Stabilising Carriers
Application:
12/543,942 →
Publication:
US 2010/0076023
Imidazo[1,2-A]Pyridines and Their Use as Pharmaceuticals
Imidazo[1,2-A]Azines and Their Use as Pharmaceuticals
Imaging probes
Bicyclic Aryl-Sulfonic Acid [1,3,4]-Thiadiazol-2-Yl-Amides, Processes for Their Preparation, Pharmaceutical Compositions and Methods for Their Use
Imidazolidine Carboxamide Derivatives as Lipase and Phospholipase Inhibitors
Use of 4 Cyclopropylmethoxy-N-(3,5 Dichloro-1 Oxido-Pyridin-4 Yl)-5-(Methoxy)Pyridine-2 Carboxamide for the Treatment of Spinal Cord Traumas
Use of 4-Cyclopropylmethoxy-N-(3,5-Dichloro-1-Oxido-4-Pyridin-4-Yl)-5-(Methoxy)Pyridine-2-Carboxamide in the Treatment of Cranial Traumas
Use of 4-Cyclopropylmethoxy-N-(3,5-Dichloro-1-Oxidopyridin-4-Yl)-5-(Methoxy)Pyridine-2-Carboxamide for the Treatment of Motor Disorders Related to Parkinson's Disease
Application:
12/573,326 →
Publication:
US 2010/0130554
5-Oxoisoxazoles as inhibitors of lipases and phospholipases
Microparticulate form of a Tetrahydropyridine derivative
Application:
12/573,455 →
Publication:
US 2010/0021541
Use of N-Heterocyclylmethylbenzamides in Therapeutics
Quinoline-Carboxamide Derivatives as P2Y12 Antagonists
Transition Metal Catalyzed Synthesis of N-Aminoindoles
2-Heteroaryl-Pyrrolo[3,4-C]Pyrrole Derivatives and Their Use as Scd Inhibitors
Arylamide Pyrimidone Derivatives
Arylamide Pyrimidone Compounds
Heteroarylamide Pyrimidone Derivatives
Heteroarylamide Pyrimidone Compounds
Method for Preparing Enantiomerically Enriched N-Carboxyanhydride
New Fluorene Derivatives, Compositions Containing the Same and Use Thereof as Inhibitors of the Protein Chaperone Hsp 90
N-Methylnaltrexone Zwitterion
Di(Hetero)Arylcyclohexane Derivatives, Their Preparation, Their Use and Pharmaceutical Compositions Comprising Them
Derivatives of 7-Alkynyl-1,8-Naphthyridones, Preparation Method Thereof and Use of Same in Therapeutics
Derivatives of 7-Alkynyl-1,8-Naphthyridones, Preparation Method Thereof and Use of Same in Therapeutics
New Compounds
Method and Intermediates for the Preparation of Derivatives of N (1-Benzhydrylazetidin-3-Yl)-N-Phenylmethylsulfonamide
Pyrrole Derivatives as P2Y12 Antagonists
Macrolactone Derivatives
Transition Metal Catalyzed Synthesis of 2H-Indazoles
Regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles
Application:
12/644,379 →
Publication:
US 2010/0216988
Regioselective copper catalyzed synthesis of benzimidazoles and azabenzimidazoles
Chemical Process
Process for the Palladium-Catalyzed Coupling of Terminal Alkynes with Heteroaryl Tosylates and Heteroaryl Benzenesulfonates
Process for the palladium-catalyzed coupling of terminal alkynes with aryl tosylates
Derivatives of Pyrazole 3,5-Carboxylates, Their Preparation and Their Application in Therapeutics
6-Cycloamino-3-(Pyrid-4-Yl)Imidazo[1,2-B]Pyridazine Derivatives, Preparation Thereof and Therapeutic Use Thereof
Novel Therapeutic Uses of Beta-3 Adrenergic Receptor Agonist Derivatives in Particular to Modulate Apoptosis
AS160-Like Protein, Test Systems, Methods and Uses Involving It for the Identification of Diabetes Type 2 Therapeutics
Application:
12/667,772 →
Publication:
US 2010/0256014
Ligand Binding Domains of Nuclear Receptors in Controllable Form and Methods Involving the Same
Application:
12/675,804 →
Publication:
US 2011/0177611
3-Methyl-2- ( (2S) -2- (4- (3-Methyl-L, 2, 4-0XADIAZ0L-5-Yl) Phenyl) Morpholino) -6- (Pyrim-Idin-4-Yl) Pyrimidin-4 (3H) -One as Tau Protein Kinase Inhibitor
6-Pyrimidinyl-Pyrimid-4-One Derivative
Use of CLEC1B for the Determination of Cardiovascular and Thrombotic Risk
Application:
12/679,547 →
Publication:
US 2010/0311053
Malonamide Derivatives with Antithrombotic Activity
6-CYCLOAMINO-3-(PYRIDAZIN-4-YL)IMIDAZO[1,2-b]PYRIDAZINE AND DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME
Cytotoxic Agents Comprising New Tomaymycin Derivatives and Their Therapeutic Use
1-Oxo-Isoindoline-4-Carboxamide and 1-Oxo-1,2,3,4-Tetrahydroisoquinoline-5-Carboxamide Derivatives, Preparation and Therapeutic Use Thereof
Derivatives of 1-Oxo-1,2-Dihydroisoquinoline-5-Carboxamides and of 4-Oxo-3,4-Dihydroquinazoline-8-Carboxamides, Preparation Thereof and Application Thereof in Therapeutics
1,2,3,4-TETRAHYDROPYRROLO[1,2-A]PYRAZINE-6-CARBOXAMIDE AND 2,3,4,5-TETRAHYDROPYRROLO[1,2-a][1,4]-DIAZEPINE-7-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF
Application:
12/693,601 →
Publication:
US 2010/0197668
Novel 6-Triazolopyridazine Sulfanyl Benzothiazole Derivatives as Met Inhibitors
4-[(Arylmethyl)Aminomethyl]Piperidine Derivatives, Their Preparation and Their Therapeutic Application
Application:
12/693,823 →
Publication:
US 2010/0240670
Caspase Imaging Probes
Application:
12/695,604 →
Publication:
US 2010/0303728
Tricyclic N-Heteroaryl-Carboxamide Derivatives, Preparation and Therapeutic Use Thereof
Derivatives of 1-Piperazine- and 1-Homopiperazine-Carboxylates, Preparation Method Thereof and Use of Same as Inhibitors of the Faah Enzyme
Novel Substituted Tetrahydronaphthalenes, Process for the Preparation Thereof and the Use Thereof as Medicaments
Azoloarine Derivatives, Method for the Production Thereof, Pharmaceuticals Containing These Compounds and the Use Thereof
Application:
12/708,179 →
Publication:
US 2010/0240580
DERIVATIVES OF IMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDES, PREPARATION METHOD THEREOF AND USE OF SAME IN THERAPEUTICS
Use of Urate Oxidase for the Treatment or Prophylaxis of Disorders or Indirect Sequelae of the Heart Caused by Ischemic or Reperfusion Events
Application:
12/715,061 →
Publication:
US 2010/0266567
(Cyclopropylphenyl)Phenyloxamides, Method for the Production Thereof, and Use of Same as a Medicament
(Carboxylalkylenephenyl)Phenyloxamides, Method for the Production Thereof and Use of Same as a Medicament
Phenothiazine Derivative Having a Double Bond, Method for the Production Thereof, and Use Thereof as a Pharmaceutical
Novel Therapeutic Uses of Adrenergic Alpha-1 Receptor Antagonists
Triazolopyridine Derivatives as Inhibitors of Lipases and Phospholipases
Application:
12/731,225 →
Publication:
US 2010/0190801
Nicotinamide Derivatives, Preparation Thereof and Therapeutic Use Thereof
Application:
12/732,749 →
Publication:
US 2010/0222319
Use of Norgestimate as a Selective Inhibitor of TRPC3, TRPC6 and TRPC7 Ion Channels
Antibodies Specific of the Beta-Amyloid Peptides and Their Uses as Diagnostic Agents or Drugs
Quinazolinedione Derivatives, Preparation Thereof and Therapeutic Uses Thereof
5,6-Diaryl Pyridines Substituted in the 2- and 3-Position, Preparation Thereof and Therapeutic Use Thereof
6-Aryl/Heteroalkyloxy Benzothiazole and Benzimidazole Derivatives, Method for Preparing Same, Application Thereof as Drugs, Pharmaceutical Compositions and Novel Use in Particular as C-Met Inhibitors
Method for the preparation of morphine compounds
N-(Heteroaryl)-1-Heteroarylalkyl-1H-Indole-2-Carboxamide Derivatives, Preparation and Therapeutic Use Thereof
Cyclic Pyridyl-N-[1,3,4]-Thiadiazol-2-Yl-Benzene Sulfonamides, Processes for Their Preparation and Their Use as Pharmaceuticals
Method for Preparing Azetidine Derivatives
Therapeutic Use of N-(Arylalkyl)-1H-Pyrrolopyridine-2-Carboxamide Derivatives
Application:
12/815,593 →
Publication:
US 2010/0249183
Process for the Preparation of 6-Substituted-1-(2H)-Isoquinolinones
Pyrazole-Carboxamide Derivatives as P2Y12 Antagonists
Heterocyclic Pyrazole-Carboxamidesas P2Y12 Antagonists
Azetidine Derivatives, Their Preparation and Their Application in Therapy
6-Heterocyclic-Imidazo[1,2-A]Pyridine-2-Carboxamide Derivatives, Preparation and Therapeutic Use Thereof
Derivatives of Dioxan-2-Alkyl Carbamates, Preparation Thereof and Application Thereof in Therapeutics
N-(Aminoheteroaryl)-1H-indole-2-carboxamide derivatives, and preparation and therapeutic application thereof
Diacyl Indazole Derivatives as Lipase and Phospholipase Inhibitors
Azabicyclic Carboxamide Derivatives, Preparation Thereof and Therapeutic Use Thereof
Bicyclic Derivatives of Azabicyclic Carboxamides, Preparation Thereof and Therapeutic Use Thereof
N-Azabicyclic Carboxamide Derivatives, Preparation Thereof and Therapeutic Use Thereof
Derivatives of Indole-2-Carboxamides and of Azaindole-2-Carboxamides Substituted with a Silanyl Group, Preparation Thereof and Therapeutic Use Thereof
Tetrahydroquinoxaline Urea Derivatives
Substituted Heteroarylamide Oxazepinopyrimidone Derivatives
Substituted Heteroarylamide Diazepinopyrimidone Derivatives
Substituted Arylamide Oxazepinopyrimidone Derivatives
Substituted Arylamide Diazepinopyrimidone Derivatives
Cyclic Indole-3-Carboxamides, Their Preparation and Their Use as Pharmaceuticals
Cyclic Azaindole-3-Carboxamides, Their Preparation and Their Use as Pharmaceuticals
Combination of a Long-Acting Hypnotic Agent and a Short-Acting Hypnotic Agent and Therapeutic Use Thereof
Application:
12/846,078 →
Publication:
US 2010/0291204
Triazolopyridazines as PAR1 Inhibitors, Production Thereof, and Use as Medicaments
Imidazopyridazines as PAR1 Inhibitors, Production Thereof, and Use as Medicaments
Triazolium Salts as PAR1 Inhibitors, Production Thereof, and Use as Medicaments
SF5 Derivatives as PAR1 Inhibitors, Production Thereof, and Use as Medicaments
Combination of a Bis-Thiazolium Salt or a Precursor Thereof and Artemisinin or a Derivative Thereof for Treating Acute Malaria
5,6-Bisaryl-2-Pyridine-Carboxamide Derivatives, Preparation Thereof and Therapeutic Application Thereof as Urotensin Ii Receptor Antagonists
Novel aromatic fluoroglycoside derivatives, pharmaceuticals comprising said compounds and the use thereof
Application:
12/851,944 →
Publication:
US 2011/0059910
Novel 3-Aminoalkyl-1,3-Dihydro-2H-Indol-2-One Derivatives, Preparation Thereof and Therapeutic Use Thereof
Chlorothiophene-Isoxazoles as Inhibitors of Coagulation Factors Xa and Thrombin
Chlorothiophene-Amides as Inhibitors of Coagulation Factors Xa and Thrombin
Covalently Binding Imaging Probes
Application:
12/860,544 →
Publication:
US 2011/0059018
Method for Preparing Combretastatin
Application:
12/869,997 →
Publication:
US 2011/0124899
Photochemical Process for Producing Artemisinin
Platinum-N-Heterocyclic Carbene Derivatives, Preparation Thereof and Therapeutic Use Thereof
Process for the Production of Artemisinin Intermediates
HSP90 Inhibitory Carbazole Derivatives, Compositions Containing Same and Use Thereof
Leptomycin Derivatives
Application:
12/881,792 →
Publication:
US 2011/0002947
Polysubstituted Derivatives of 2-Aryl-6-Phenyl-Imidazo[1,2-a]Pyridines, and Preparation and Therapeutic Use Thereof
Polysubstituted Derivatives of 2-Heteroaryl-6-Phenylimidazo[1,2-a]Pyridines, and Preparation and Therapeutic Use Thereof
Polysubstituted Derivatives of 6-Heteroarylimidazo[1,2-a]Pyridines, and Preparation and Therapeutic Use Thereof
Polysubstituted 2-Aryl-6-Phenylimidazo[1,2-a]Pyridine Derivatives, and Preparation and Therapeutic Use Thereof
Highly Bridged Peptides from Actinomadura Namibiensis
Application:
12/895,106 →
Publication:
US 2011/0144001
Tetrahydroisoquinoline Sulfonamide Derivatives, the Preparation Thereof, and the Use of the Same in Therapeutics
Combination of Dronedarone with at Least One Diuretic, and Therapeutic Use Thereof
Application:
12/903,374 →
Publication:
US 2011/0136899
Use of Dronedarone or a Pharmaceutically Acceptable Salt Thereof, for the Preparation of a Medicament for Regulating the Potasium Level in the Blood
Application:
12/903,377 →
Publication:
US 2011/0124724
1,3-Dihydro-2H-Pyrrolo[3,2-B]Pyridin-2-One Derivatives, Preparation Thereof and Therapeutic Uses Thereof
Azolopyridin-2-One Derivatives as Lipase and Phospholipase Inhibitors
Application:
12/914,045 →
Publication:
US 2011/0039883
Fluorescence Based Assay to Detect Sodium/Calcium Exchanger (Ncx ) "Reverse Mode" Modulating Compounds
Application:
12/922,741 →
Publication:
US 2011/0124033
Fluorescence Based Assay to Detect Sodium/Calcium Exchanger "Forward Mode" Modulating Compounds
Application:
12/922,749 →
Publication:
US 2011/0117574
Cathepsin C-Based Screening Methods for Identifying Modulators of Pain
Pyrrole Derivatives, Their Preparation and Their Therapeutic Application
Use of Dronedarone for the Preparation of a Medicament for Use in the Prevention of Cardiovascular Hospitalization or of Mortality
Application:
12/951,471 →
Publication:
US 2011/0224293
Use of Dronedarone for the Preparation of a Medicament for Use in the Prevention of Cardiovascular Hospitalization or of Mortality
Application:
12/951,494 →
Publication:
US 2011/0213027
Derivatives of 5-Pyridinyl-1-Azabicyclo[3.2.1]Octane, Preparation Method Thereof and Use of Same in Therapeutics
Fumarate Salt of 4-Bromophenyl 1,4-Diazabicyclo[3.2.2]Nonane-4-Carboxylate, Crystalline Forms Thereof, Preparation Thereof and Therapeutic Use Thereof
Combination of a Nicotinic Receptor Partial Agonist and of an Acetylcholinesterase Inhibitor, Pharmaceutical Composition Containing Same and Use Thereof in the Treatment of Cognitive Disorders
Application:
12/958,025 →
Publication:
US 2011/0136791
Dronedarone for the Prevention of Permanent Atrial Fibrillation
Application:
12/962,102 →
Publication:
US 2011/0166220
Use of Dronedarone for the Preparation of a Medicament for Use in the Prevention of Cardioversion
Application:
12/962,115 →
Publication:
US 2011/0166221
Derivatives of (Bridged Piperazinyl)-1-Alkanone and Use Thereof as P75 Inhibitors
Filling Structure for a Graft System and Methods of Use
Application:
12/966,852 →
Publication:
US 2011/0276078
Substituted Alkyl Pyrimidin-4-One Derivatives
Substituted Pyrimidone Derivatives
Substituted Tricyclic Derivatives
Substituted Triazinone Derivatives
Substituted Pyrimido Isoquinoline Derivatives
Substituted N-Oxide Pyrazine Derivatives
6-Substituted Isoquinolines and Isoquinolinones
Novel Derivatives of Pyrroloindole Which Are Inhibitors of HSP90, Compositions Containing Same, and Use Thereof
Pyridinopyridinone Derivatives, Preparation Thereof and Therapeutic Use Thereof
Substituted 1-Benzyl-Cinnolin-4(1H)-One Derivatives, Preparation Thereof, and Therapeutic Use Thereof
Use of GPR151 Modulators for the Treatment of Pain
Application:
12/993,024 →
Publication:
US 2011/0177096
Macrocyclic Urea and Sulfamide Derivatives as Inhibitors of Tafia
Annelated Pyrrolidin Sulfonamides with Oxadiazolone Headgroup, Processes for Their Preparation and Their Use as Pharmaceuticals
Sulfonamides with Heterocycle and Oxadiazolone Headgroup, Processes for Their Preparation and Their Use as Pharmaceuticals
Azacarboline Derivatives, Preparation Method Thereof and Therapeutic Use of Same
Application:
12/997,326 →
Publication:
US 2011/0178053
Bi- and Polycyclic Substituted Isoquinoline and Isoquinolinone Derivatives
Substituted Isoquinolines and Isoquinolinones as Rho Kinase Inhibitors
Fgf-R4 Receptor-Specific Antagonists
Application:
13/002,845 →
Publication:
US 2011/0150903
Heterocyclic Compounds, Processes for Their Preparation, Medicaments Comprising These Compounds, and the Use Thereof
Oxazolopyrimidines as Edg-1 Receptor Agonists
Novel Imidazo[1,2-a]Pyridine Derivatives, Method for the Preparation Thereof, Use Thereof as Medicaments, Pharmaceutical Compositions and Novel Use in Particular as Met Inhibitors
Application:
13/003,604 →
Publication:
US 2011/0257171
Use of Idrabiotaparinux for Decreasing the Incidence of Bleedings During an Antithrombotic Treatment
Application:
13/003,623 →
Publication:
US 2011/0245200
Alkylthiazol Carbamate Derivatives, Preparation Thereof and Therapeutic Use Thereof
NOVEL IMIDAZO[1,2-a]PYRIMIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE, IN PARTICULAR AS MET INHIBITORS
Application:
13/007,830 →
Publication:
US 2011/0263593
Carbamoylbenzotriazole Derivatives as Inhibitors of Lipases and Phospholipases
Application:
13/009,951 →
Publication:
US 2011/0118321
Indol-2-One Derivatives Disubstituted in the 3-Position, Preparation Thereof and Therapeutic Use Thereof
Pyrrolidinyl-Alkyl-Amide Derivatives, Their Preparation, and Their Therapeutic Application as CCR3 Receptor Ligands
EGLN2 Variants and Use Thereof in Preventing or Treating Thromboembolic Disorders and Coronary Heart Diseases
Novel imidazo[1,5-a]pyridine derivatives, method for preparing same and pharmaceutical compositions containing same
Use of Dronedarone for the Preparation of a Medicament for the Prevention of Stroke or Transient Ischemic Attack
Application:
13/020,889 →
Publication:
US 2011/0230552
Novel Triazolo(4,3-a)Pyridine Derivatives, Process for the Preparation Thereof, Use Thereof as Medicaments, Pharmaceutical Compositions and Novel Use, in Particular as Met Inhibitors
Application:
13/054,663 →
Publication:
US 2011/0263594
Streptospirole Derivatives
Thiophene-2-Carboxamide Derivatives, Preparation Thereof and Therapeutic Use Thereof
NEW COMBINATION OF ACTIVE INGREDIENTS CONTAINING AN a1-ANTAGONIST AND A PDE 4 INHIBITOR
Application:
13/059,760 →
Publication:
US 2011/0263621
Polysaccharides with Antithrombotic Activity, Including a Covalent Bond and an Amino Chain
Substituted Aminoindanes and Analogs Thereof, and the Pharmaceutical Use Thereof
2-Heteroaryl-Pyrrolo [3,4-C]Pyrrole Derivatives, and Use Thereof as Scd Inhibitors
Methods for Determining Sodium-Proton-Exchanger Ligand Efficiency
Novel Anti-CD38 Antibodies for the Treatment of Cancer
Application:
13/069,705 →
Publication:
US 2011/0262454
Method for Preparing 1,6:2,3-Dianhydro-Beta-D-Mannopyranose
Short Synthetic Pathway for 1,6:2,3-Dianhydro-Beta-D-Mannopyranose
Tropane Urea Derivatives, Preparation Thereof and Therapeutic Application Thereof as Modulators of the Activity of 11BETAHSD1
Use of 7-Chloro-N,N,5-Trimethyl-4-Oxo-3-Phenyl-3,5-Dihydro-4H-Pyridazino[4,5-B] Indole-1-Acetamide as a Biomarker of Peripheral Benzodiazepine Receptor Levels
Application:
13/126,648 →
Publication:
US 2012/0039816
Use of Inhibitors of PLAC8 Activity for the Modulation of Adipogenesis
Application:
13/127,841 →
Publication:
US 2012/0035241
Method for Preparing Eplivanserin Hemifumarate
Application:
13/128,756 →
Publication:
US 2012/0022292
6-Cycloamino-3-(1H-Pyrrolo[2,3-B]Pyridin-4-Yl)Imidazo[1,2-B]Pyridazine Derivatives, Preparation Thereof and Therapeutic Use Thereof
Method of Treating Sleep Disorders Using Eplivanserin
Application:
13/129,019 →
Publication:
US 2012/0108669
Carbamate Derivatives of Alkyl-Heterocycles, Preparation Thereof and Therapeutic Use Thereof
Antitumor Combinations Containing Antibodies Recognizing Specifically CD38 and Melphalan
Antitumor Combinations Containing Antibodies Recognizing Specifically CD38 and Vincristine
Antitumor Combinations Containing Antibodies Recognizing Specifically CD38 and Cytarabine
Application:
13/130,867 →
Publication:
US 2012/0093806
Antitumor Combinations Containing Antibodies Recognizing Specifically CD38 and Cyclophosphamide
Application:
13/131,389 →
Publication:
US 2011/0305690
Method of Screening a Modulator of Endothelial No Synthase Comprising the Use of Heme Binding Protein 1
Macrolactone Derivatives, Method for the Production Thereof and Use Thereof for the Treatment of Cancer
Application:
13/139,458 →
Publication:
US 2011/0306563
DERIVATIVES OF 6-CYCLOAMINO-2-THIENYL-3-(PYRIDIN-4-YL)IMIDAZO[1,2-b]-PYRIDAZINE AND 6-CYCLOAMINO-2-FURANYL-3-(PYRIDIN-4-YL)IMIDAZO[1,2-b]-PYRIDAZINE, PREPARATION AND THERAPEUTIC USE THEREOF
Application:
13/141,006 →
Publication:
US 2013/0190314
Substituted Pyrazoles, Compositions Containing These, Method of Production and Use
Substituted Pyrazoles, Compositions Containing These, Method of Production and Use
Isoquinoline Derivatives
Cyclohexylamine Isoquinolone Derivatives
Methods for Reducing Risk
Application:
13/211,673 →
Publication:
US 2011/0297563
Topical Skin Treatment Kits
Application:
13/213,471 →
Publication:
US 2011/0306566
Triazolopyridazines as PAR1 Inhibitors, Production Thereof, and Use as Medicaments
Spirocyclic nitriles as protease inhibitors
1-Pyrazolo[4,3-C]Isoquinoline Derivatives, Preparation Thereof and Therapeutic Use Thereof
Substituted N-Phenyl-Bipyrrolidine Carboxamides and Therapeutic Use Thereof
EGLN2 Variants and Use Thereof in Preventing or Treating Thromboembolic Disorders and Coronary Heart Diseases
2H or 3H-Benzo[E]Indazol-1-Yl Carbamate Derivatives, the Preparation and Therapeutic Use Thereof
Tricyclic N-Heteroaryl-Carboxamide Derivatives Containing a Benzimidazole Unit, Method for Preparing Same and Their Therapeutic Use
Novel Anti-CD38 Antibodies for the Treatment of Cancer
Application:
13/372,770 →
Publication:
US 2012/0156218
Disubstituted [4-(5-Aminomethyl-Phenyl)-Piperidin-1-Yl]- 1H-Indol-3-Yl]-Methanones
Application:
13/396,111 →
Publication:
US 2012/0142735
Method for Preparing Enantiomerically Enriched N-Carboxyanhydride
Application:
13/399,337 →
Publication:
US 2012/0215007
Substituted Dihydro Benzocycloalkyloxymethyl Oxazolopyrimidinones, Preparation and Use Thereof
Azabicycloalkane Derivatives, Preparation Thereof and Use Thereof in Therapy
Phenyloxadiazole Derivatives as Pgds Inhibitors
Related Assignments
(1)
Other recorded transfers of the patents in this record — the chain of ownership.